Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | PIM3 | 2.8 | 1000 | nM |
Abemaciclib | DYRK2 | 2.8 | 100 | nM |
Abemaciclib | DAPK3 | 2.9 | 1000 | nM |
Abemaciclib | PIM1 | 2.9 | 1000 | nM |
Abemaciclib | ROCK2 | 3.0 | 1000 | nM |
Abemaciclib | CDKL3 | 3.1 | 1000 | nM |
Abemaciclib | NEK10 | 3.5 | 100 | nM |
Abemaciclib | HIPK1 | 3.7 | 100 | nM |
Abemaciclib | JNK1 | 4.0 | 1000 | nM |
Abemaciclib | FLT3(D835V) | 4.0 | 1000 | nM |
Abemaciclib | JNK3 | 4.0 | 1000 | nM |
Abemaciclib | KPCE | 4.1 | 1000 | nM |
Abemaciclib | CDK4-cyclinD1 | 4.1 | 1000 | nM |
Abemaciclib | CAMK2A | 4.1 | 100 | nM |
Abemaciclib | PCTK2 | 4.3 | 1000 | nM |
Abemaciclib | CAMK2B | 4.5 | 100 | nM |
Abemaciclib | PIM1 | 4.7 | 100 | nM |
Abemaciclib | TAK1 | 4.7 | 1000 | nM |
Abemaciclib | CAMKK2 | 4.7 | 1000 | nM |
Abemaciclib | DCAMKL3 | 4.8 | 1000 | nM |
Abemaciclib | RPS6KA4(Kin.Dom.2-C-terminal) | 4.9 | 1000 | nM |
Abemaciclib | FLT3(ITD,D835V) | 5.1 | 1000 | nM |
Abemaciclib | PIM3 | 5.2 | 100 | nM |
Abemaciclib | ROCK1 | 5.2 | 1000 | nM |
Abemaciclib | FYV1 | 5.5 | 1000 | nM |