Abemaciclib KINOMEscan - Dataset (ID:20338)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | DYRK1B | 0.8 | 1000 | nM |
Abemaciclib | SGK1 | 0.8 | 1000 | nM |
Abemaciclib | DYRK2 | 0.9 | 1000 | nM |
Abemaciclib | CDKL2 | 0.9 | 1000 | nM |
Abemaciclib | IRAK1 | 0.9 | 100 | nM |
Abemaciclib | CDKL5 | 0.9 | 100 | nM |
Abemaciclib | CLK1 | 1.0 | 1000 | nM |
Abemaciclib | DYRK1B | 1.0 | 100 | nM |
Abemaciclib | ERK8 | 1.1 | 100 | nM |
Abemaciclib | CSNK2A1 | 1.2 | 1000 | nM |
Abemaciclib | YSK4 | 1.2 | 1000 | nM |
Abemaciclib | GSK3B | 1.2 | 1000 | nM |
Abemaciclib | TAOK3 | 1.4 | 1000 | nM |
Abemaciclib | DRAK1 | 1.4 | 1000 | nM |
Abemaciclib | CDK7 | 1.7 | 1000 | nM |
Abemaciclib | SGK3 | 1.8 | 1000 | nM |
Abemaciclib | JAK3(JH1domain-catalytic) | 1.8 | 1000 | nM |
Abemaciclib | GCN2(Kin.Dom.2,S808G) | 1.9 | 1000 | nM |
Abemaciclib | ICK | 1.9 | 1000 | nM |
Abemaciclib | AAK1 | 2.0 | 1000 | nM |
Abemaciclib | CSNK2A1 | 2.3 | 100 | nM |
Abemaciclib | DYRK1A | 2.3 | 100 | nM |
Abemaciclib | STK16 | 2.6 | 1000 | nM |
Abemaciclib | CSNK2A2 | 2.6 | 100 | nM |
Abemaciclib | SGK2 | 2.7 | 1000 | nM |