Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | MAP3K1 | 73.0 | 100 | nM |
Abemaciclib | MAP3K14 | 74.0 | 1000 | nM |
Abemaciclib | BIKE | 74.0 | 100 | nM |
Abemaciclib | KPCD2 | 74.0 | 100 | nM |
Abemaciclib | NDR1 | 74.0 | 1000 | nM |
Abemaciclib | FLT3(K663Q) | 74.0 | 1000 | nM |
Abemaciclib | PKN1 | 74.0 | 100 | nM |
Abemaciclib | MINK | 75.0 | 100 | nM |
Abemaciclib | CDK9 | 75.0 | 100 | nM |
Abemaciclib | MK13 | 75.0 | 100 | nM |
Abemaciclib | M3K6 | 75.0 | 100 | nM |
Abemaciclib | RSK4(Kin.Dom.2-C-terminal) | 75.0 | 100 | nM |
Abemaciclib | EGFR(L861Q) | 75.0 | 1000 | nM |
Abemaciclib | CASK | 75.0 | 100 | nM |
Abemaciclib | EGFR(E746-A750del) | 76.0 | 1000 | nM |
Abemaciclib | DAPK1 | 76.0 | 100 | nM |
Abemaciclib | PHKG1 | 76.0 | 100 | nM |
Abemaciclib | NEK1 | 76.0 | 100 | nM |
Abemaciclib | FLT3-autoinhibited | 76.0 | 100 | nM |
Abemaciclib | MAP4K5 | 76.0 | 1000 | nM |
Abemaciclib | MRCKA | 76.0 | 1000 | nM |
Abemaciclib | KPCI | 77.0 | 1000 | nM |
Abemaciclib | RSK3(Kin.Dom.2-C-terminal) | 77.0 | 100 | nM |
Abemaciclib | MET(M1250T) | 77.0 | 100 | nM |
Abemaciclib | LOK | 78.0 | 1000 | nM |