Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small Molecule Protein % Control Assay compound conc Conc unit
Abemaciclib MAP3K1 73.0 100
nM
Abemaciclib MAP3K14 74.0 1000
nM
Abemaciclib BIKE 74.0 100
nM
Abemaciclib KPCD2 74.0 100
nM
Abemaciclib NDR1 74.0 1000
nM
Abemaciclib FLT3(K663Q) 74.0 1000
nM
Abemaciclib PKN1 74.0 100
nM
Abemaciclib MINK 75.0 100
nM
Abemaciclib CDK9 75.0 100
nM
Abemaciclib MK13 75.0 100
nM
Abemaciclib M3K6 75.0 100
nM
Abemaciclib RSK4(Kin.Dom.2-C-terminal) 75.0 100
nM
Abemaciclib EGFR(L861Q) 75.0 1000
nM
Abemaciclib CASK 75.0 100
nM
Abemaciclib EGFR(E746-A750del) 76.0 1000
nM
Abemaciclib DAPK1 76.0 100
nM
Abemaciclib PHKG1 76.0 100
nM
Abemaciclib NEK1 76.0 100
nM
Abemaciclib FLT3-autoinhibited 76.0 100
nM
Abemaciclib MAP4K5 76.0 1000
nM
Abemaciclib MRCKA 76.0 1000
nM
Abemaciclib KPCI 77.0 1000
nM
Abemaciclib RSK3(Kin.Dom.2-C-terminal) 77.0 100
nM
Abemaciclib MET(M1250T) 77.0 100
nM
Abemaciclib LOK 78.0 1000
nM