Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small Molecule Protein % Control Assay compound conc Conc unit
Abemaciclib ABL1(H396P)-nonphosphorylated 80.0 100
nM
Abemaciclib AKT3 100.0 100
nM
Abemaciclib ABL1(Y253F)-phosphorylated 100.0 100
nM
Abemaciclib ALK 78.0 100
nM
Abemaciclib ABL1(F317I)-phosphorylated 91.0 100
nM
Abemaciclib ALK(C1156Y) 81.0 100
nM
Abemaciclib ABL1-nonphosphorylated 92.0 100
nM
Abemaciclib ALK(L1196M) 78.0 100
nM
Abemaciclib ABL1(H396P)-phosphorylated 89.0 100
nM
Abemaciclib AMPK-alpha1 80.0 100
nM
Abemaciclib ABL1-phosphorylated 98.0 100
nM
Abemaciclib AMPK-alpha2 100.0 100
nM
Abemaciclib AAK1 20.0 100
nM
Abemaciclib ANKK1 100.0 100
nM
Abemaciclib ABL2 95.0 100
nM
Abemaciclib NUAK1 98.0 100
nM
Abemaciclib ABL1(M351T)-phosphorylated 100.0 100
nM
Abemaciclib M3K5 100.0 100
nM
Abemaciclib ACVR1 100.0 100
nM
Abemaciclib M3K6 75.0 100
nM
Abemaciclib ABL1(F317L)-nonphosphorylated 99.0 100
nM
Abemaciclib AURKA 100.0 100
nM
Abemaciclib ACVR1B 100.0 100
nM
Abemaciclib AURKB 92.0 100
nM
Abemaciclib CDK5 100.0 100
nM