Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | EPHA8 | 97.0 | 100 | nM |
Abemaciclib | CDK2 | 94.0 | 100 | nM |
Abemaciclib | EPHB1 | 92.0 | 100 | nM |
Abemaciclib | ACVR1 | 100.0 | 100 | nM |
Abemaciclib | EPHB2 | 95.0 | 100 | nM |
Abemaciclib | CDK3 | 100.0 | 100 | nM |
Abemaciclib | EPHB3 | 93.0 | 100 | nM |
Abemaciclib | M3K6 | 75.0 | 100 | nM |
Abemaciclib | EPHB4 | 85.0 | 100 | nM |
Abemaciclib | CDK4-cyclinD1 | 54.0 | 100 | nM |
Abemaciclib | EPHB6 | 100.0 | 100 | nM |
Abemaciclib | ABL1(F317L)-nonphosphorylated | 99.0 | 100 | nM |
Abemaciclib | ERBB2 | 100.0 | 100 | nM |
Abemaciclib | CDK4-cyclinD1 | 0.6 | 100 | nM |
Abemaciclib | ERBB3 | 98.0 | 100 | nM |
Abemaciclib | AURKA | 100.0 | 100 | nM |
Abemaciclib | ERBB4 | 100.0 | 100 | nM |
Abemaciclib | CDK4-cyclinD3 | 0.5 | 100 | nM |
Abemaciclib | MK03 | 100.0 | 100 | nM |
Abemaciclib | ACVR1B | 100.0 | 100 | nM |
Abemaciclib | MK01 | 100.0 | 100 | nM |
Abemaciclib | CDK5 | 100.0 | 100 | nM |
Abemaciclib | ERK3 | 100.0 | 100 | nM |
Abemaciclib | AURKB | 92.0 | 100 | nM |
Abemaciclib | OSR1 | 100.0 | 100 | nM |