Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small Molecule Protein % Control Assay compound conc Conc unit
Abemaciclib EPHA8 97.0 100
nM
Abemaciclib CDK2 94.0 100
nM
Abemaciclib EPHB1 92.0 100
nM
Abemaciclib ACVR1 100.0 100
nM
Abemaciclib EPHB2 95.0 100
nM
Abemaciclib CDK3 100.0 100
nM
Abemaciclib EPHB3 93.0 100
nM
Abemaciclib M3K6 75.0 100
nM
Abemaciclib EPHB4 85.0 100
nM
Abemaciclib CDK4-cyclinD1 54.0 100
nM
Abemaciclib EPHB6 100.0 100
nM
Abemaciclib ABL1(F317L)-nonphosphorylated 99.0 100
nM
Abemaciclib ERBB2 100.0 100
nM
Abemaciclib CDK4-cyclinD1 0.6 100
nM
Abemaciclib ERBB3 98.0 100
nM
Abemaciclib AURKA 100.0 100
nM
Abemaciclib ERBB4 100.0 100
nM
Abemaciclib CDK4-cyclinD3 0.5 100
nM
Abemaciclib MK03 100.0 100
nM
Abemaciclib ACVR1B 100.0 100
nM
Abemaciclib MK01 100.0 100
nM
Abemaciclib CDK5 100.0 100
nM
Abemaciclib ERK3 100.0 100
nM
Abemaciclib AURKB 92.0 100
nM
Abemaciclib OSR1 100.0 100
nM