Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | AMPK-alpha2 | 100.0 | 100 | nM |
Abemaciclib | EGFR(L858R,T790M) | 83.0 | 100 | nM |
Abemaciclib | CAMKK2 | 42.0 | 100 | nM |
Abemaciclib | EGFR(L861Q) | 87.0 | 100 | nM |
Abemaciclib | AAK1 | 20.0 | 100 | nM |
Abemaciclib | EGFR(S752-I759del) | 100.0 | 100 | nM |
Abemaciclib | CASK | 75.0 | 100 | nM |
Abemaciclib | EGFR(T790M) | 98.0 | 100 | nM |
Abemaciclib | ANKK1 | 100.0 | 100 | nM |
Abemaciclib | EIF2AK1 | 97.0 | 100 | nM |
Abemaciclib | CDC2L1 | 100.0 | 100 | nM |
Abemaciclib | EPHA1 | 100.0 | 100 | nM |
Abemaciclib | ABL2 | 95.0 | 100 | nM |
Abemaciclib | EPHA2 | 91.0 | 100 | nM |
Abemaciclib | CDC2L2 | 100.0 | 100 | nM |
Abemaciclib | EPHA3 | 100.0 | 100 | nM |
Abemaciclib | NUAK1 | 98.0 | 100 | nM |
Abemaciclib | EPHA4 | 99.0 | 100 | nM |
Abemaciclib | CDC2L5 | 63.0 | 100 | nM |
Abemaciclib | EPHA5 | 99.0 | 100 | nM |
Abemaciclib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Abemaciclib | EPHA6 | 95.0 | 100 | nM |
Abemaciclib | CDK11 | 100.0 | 100 | nM |
Abemaciclib | EPHA7 | 97.0 | 100 | nM |
Abemaciclib | MST2 | 73.0 | 100 | nM |