Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small Molecule Protein % Control Assay compound conc Conc unit
Abemaciclib DRAK1 68.0 100
nM
Abemaciclib ALK(C1156Y) 81.0 100
nM
Abemaciclib DRAK2 88.0 100
nM
Abemaciclib CAMK2A 4.1 100
nM
Abemaciclib DYRK1A 2.3 100
nM
Abemaciclib ABL1-nonphosphorylated 92.0 100
nM
Abemaciclib DYRK1B 1.0 100
nM
Abemaciclib CAMK2B 4.5 100
nM
Abemaciclib DYRK2 2.8 100
nM
Abemaciclib ALK(L1196M) 78.0 100
nM
Abemaciclib EGFR 100.0 100
nM
Abemaciclib KCC2D 6.1 100
nM
Abemaciclib EGFR(E746-A750del) 92.0 100
nM
Abemaciclib ABL1(H396P)-phosphorylated 89.0 100
nM
Abemaciclib EGFR(G719C) 86.0 100
nM
Abemaciclib CAMK2G 8.9 100
nM
Abemaciclib EGFR(G719S) 89.0 100
nM
Abemaciclib AMPK-alpha1 80.0 100
nM
Abemaciclib EGFR(L747-E749del, A750P) 100.0 100
nM
Abemaciclib KCC4 100.0 100
nM
Abemaciclib EGFR(L747-S752del, P753S) 88.0 100
nM
Abemaciclib ABL1-phosphorylated 98.0 100
nM
Abemaciclib EGFR(L747-T751del,Sins) 89.0 100
nM
Abemaciclib KKCC1 71.0 100
nM
Abemaciclib MARK4 100.0 100
nM