Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | DRAK1 | 68.0 | 100 | nM |
Abemaciclib | ALK(C1156Y) | 81.0 | 100 | nM |
Abemaciclib | DRAK2 | 88.0 | 100 | nM |
Abemaciclib | CAMK2A | 4.1 | 100 | nM |
Abemaciclib | DYRK1A | 2.3 | 100 | nM |
Abemaciclib | ABL1-nonphosphorylated | 92.0 | 100 | nM |
Abemaciclib | DYRK1B | 1.0 | 100 | nM |
Abemaciclib | CAMK2B | 4.5 | 100 | nM |
Abemaciclib | DYRK2 | 2.8 | 100 | nM |
Abemaciclib | ALK(L1196M) | 78.0 | 100 | nM |
Abemaciclib | EGFR | 100.0 | 100 | nM |
Abemaciclib | KCC2D | 6.1 | 100 | nM |
Abemaciclib | EGFR(E746-A750del) | 92.0 | 100 | nM |
Abemaciclib | ABL1(H396P)-phosphorylated | 89.0 | 100 | nM |
Abemaciclib | EGFR(G719C) | 86.0 | 100 | nM |
Abemaciclib | CAMK2G | 8.9 | 100 | nM |
Abemaciclib | EGFR(G719S) | 89.0 | 100 | nM |
Abemaciclib | AMPK-alpha1 | 80.0 | 100 | nM |
Abemaciclib | EGFR(L747-E749del, A750P) | 100.0 | 100 | nM |
Abemaciclib | KCC4 | 100.0 | 100 | nM |
Abemaciclib | EGFR(L747-S752del, P753S) | 88.0 | 100 | nM |
Abemaciclib | ABL1-phosphorylated | 98.0 | 100 | nM |
Abemaciclib | EGFR(L747-T751del,Sins) | 89.0 | 100 | nM |
Abemaciclib | KKCC1 | 71.0 | 100 | nM |
Abemaciclib | MARK4 | 100.0 | 100 | nM |