Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | WEE1 | 94.0 | 1000 | nM |
Abemaciclib | VRK2 | 94.0 | 1000 | nM |
Abemaciclib | VRK2 | 100.0 | 100 | nM |
Abemaciclib | VGFR2 | 100.0 | 1000 | nM |
Abemaciclib | VGFR2 | 79.0 | 100 | nM |
Abemaciclib | VGFR1 | 95.0 | 100 | nM |
Abemaciclib | VGFR1 | 87.0 | 1000 | nM |
Abemaciclib | ULK3 | 35.0 | 1000 | nM |
Abemaciclib | ULK3 | 83.0 | 100 | nM |
Abemaciclib | ULK2 | 31.0 | 1000 | nM |
Abemaciclib | ULK2 | 83.0 | 100 | nM |
Abemaciclib | ULK1 | 48.0 | 1000 | nM |
Abemaciclib | ULK1 | 100.0 | 100 | nM |
Abemaciclib | TYRO3 | 97.0 | 100 | nM |
Abemaciclib | TYRO3 | 81.0 | 1000 | nM |
Abemaciclib | TYK2(JH2domain-pseudokinase) | 100.0 | 100 | nM |
Abemaciclib | TYK2(JH2domain-pseudokinase) | 91.0 | 1000 | nM |
Abemaciclib | TYK2(JH1domain-catalytic) | 92.0 | 1000 | nM |
Abemaciclib | TYK2(JH1domain-catalytic) | 100.0 | 100 | nM |
Abemaciclib | TXK | 100.0 | 100 | nM |
Abemaciclib | TXK | 100.0 | 1000 | nM |
Abemaciclib | TTK | 47.0 | 1000 | nM |
Abemaciclib | TTK | 62.0 | 100 | nM |
Abemaciclib | TSSK3 | 100.0 | 100 | nM |
Abemaciclib | TSSK3 | 82.0 | 1000 | nM |