Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small Molecule Protein % Control Assay compound conc Conc unit
Abemaciclib WEE1 94.0 1000
nM
Abemaciclib VRK2 94.0 1000
nM
Abemaciclib VRK2 100.0 100
nM
Abemaciclib VGFR2 100.0 1000
nM
Abemaciclib VGFR2 79.0 100
nM
Abemaciclib VGFR1 95.0 100
nM
Abemaciclib VGFR1 87.0 1000
nM
Abemaciclib ULK3 35.0 1000
nM
Abemaciclib ULK3 83.0 100
nM
Abemaciclib ULK2 31.0 1000
nM
Abemaciclib ULK2 83.0 100
nM
Abemaciclib ULK1 48.0 1000
nM
Abemaciclib ULK1 100.0 100
nM
Abemaciclib TYRO3 97.0 100
nM
Abemaciclib TYRO3 81.0 1000
nM
Abemaciclib TYK2(JH2domain-pseudokinase) 100.0 100
nM
Abemaciclib TYK2(JH2domain-pseudokinase) 91.0 1000
nM
Abemaciclib TYK2(JH1domain-catalytic) 92.0 1000
nM
Abemaciclib TYK2(JH1domain-catalytic) 100.0 100
nM
Abemaciclib TXK 100.0 100
nM
Abemaciclib TXK 100.0 1000
nM
Abemaciclib TTK 47.0 1000
nM
Abemaciclib TTK 62.0 100
nM
Abemaciclib TSSK3 100.0 100
nM
Abemaciclib TSSK3 82.0 1000
nM