Abemaciclib KINOMEscan - Dataset (ID:20338)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | PIK3CA(H1047L) | 100.0 | 100 | nM |
Abemaciclib | PIK3CA(H1047L) | 100.0 | 1000 | nM |
Abemaciclib | PIK3CA(E545K) | 79.0 | 100 | nM |
Abemaciclib | PIK3CA(E545K) | 98.0 | 1000 | nM |
Abemaciclib | PIK3CA(E545A) | 95.0 | 100 | nM |
Abemaciclib | PIK3CA(E545A) | 100.0 | 1000 | nM |
Abemaciclib | PIK3CA(E542K) | 98.0 | 100 | nM |
Abemaciclib | PIK3CA(E542K) | 100.0 | 1000 | nM |
Abemaciclib | PIK3CA(C420R) | 100.0 | 1000 | nM |
Abemaciclib | PIK3CA(C420R) | 100.0 | 100 | nM |
Abemaciclib | PIK3CA | 100.0 | 1000 | nM |
Abemaciclib | PIK3CA | 100.0 | 100 | nM |
Abemaciclib | PIK3C3 | 12.0 | 1000 | nM |
Abemaciclib | PIK3C3 | 67.0 | 100 | nM |
Abemaciclib | PIK3C2G | 81.0 | 100 | nM |
Abemaciclib | PIK3C2G | 97.0 | 1000 | nM |
Abemaciclib | PIK3C2B | 100.0 | 100 | nM |
Abemaciclib | PIK3C2B | 100.0 | 1000 | nM |
Abemaciclib | PI42C | 65.0 | 100 | nM |
Abemaciclib | PI42C | 13.0 | 1000 | nM |
Abemaciclib | PHKG2 | 51.0 | 100 | nM |
Abemaciclib | PHKG2 | 23.0 | 1000 | nM |
Abemaciclib | PHKG1 | 76.0 | 100 | nM |
Abemaciclib | PHKG1 | 18.0 | 1000 | nM |
Abemaciclib | PGFRB | 99.0 | 100 | nM |