Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | AKT2 | 100.0 | 1000 | nM |
Abemaciclib | AKT3 | 100.0 | 100 | nM |
Abemaciclib | AKT3 | 100.0 | 1000 | nM |
Abemaciclib | ABL1(Y253F)-phosphorylated | 100.0 | 100 | nM |
Abemaciclib | ABL1(Y253F)-phosphorylated | 100.0 | 1000 | nM |
Abemaciclib | PTK6 | 100.0 | 1000 | nM |
Abemaciclib | BTK | 100.0 | 1000 | nM |
Abemaciclib | BLK | 100.0 | 100 | nM |
Abemaciclib | PTK6 | 100.0 | 100 | nM |
Abemaciclib | CDK11 | 100.0 | 1000 | nM |
Abemaciclib | BRSK2 | 100.0 | 100 | nM |
Abemaciclib | AMPK-alpha2 | 100.0 | 100 | nM |
Abemaciclib | ABL1(F317I)-phosphorylated | 100.0 | 1000 | nM |
Abemaciclib | ANKK1 | 100.0 | 100 | nM |
Abemaciclib | ANKK1 | 100.0 | 1000 | nM |
Abemaciclib | CDK5 | 100.0 | 100 | nM |
Abemaciclib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Abemaciclib | M3K5 | 100.0 | 100 | nM |
Abemaciclib | M3K5 | 100.0 | 1000 | nM |
Abemaciclib | ACVR1 | 100.0 | 100 | nM |
Abemaciclib | ABL1(M351T)-phosphorylated | 100.0 | 1000 | nM |
Abemaciclib | AURKA | 100.0 | 100 | nM |
Abemaciclib | ACVR1B | 100.0 | 100 | nM |
Abemaciclib | EPHA3 | 100.0 | 1000 | nM |
Abemaciclib | EPHA3 | 100.0 | 100 | nM |