Abemaciclib KINOMEscan - Dataset (ID:20338)

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Small Molecule Protein % Control Assay compound conc Conc unit
Abemaciclib ABL1(Y253F)-phosphorylated 100.0 100
nM
Abemaciclib ABL1(Y253F)-phosphorylated 100.0 1000
nM
Abemaciclib M3K5 100.0 1000
nM
Abemaciclib AMPK-alpha2 100.0 100
nM
Abemaciclib BMPR1A 100.0 100
nM
Abemaciclib ABL1(F317I)-phosphorylated 100.0 1000
nM
Abemaciclib BLK 100.0 100
nM
Abemaciclib ABL1(M351T)-phosphorylated 100.0 100
nM
Abemaciclib ACVR1 100.0 100
nM
Abemaciclib ABL1(M351T)-phosphorylated 100.0 1000
nM
Abemaciclib ACVR1B 100.0 100
nM
Abemaciclib ACVR1B 100.0 1000
nM
Abemaciclib BMX 100.0 1000
nM
Abemaciclib ABL1(F317I)-nonphosphorylated 100.0 100
nM
Abemaciclib ANKK1 100.0 1000
nM
Abemaciclib ACVR2B 100.0 1000
nM
Abemaciclib ACVRL1 100.0 100
nM
Abemaciclib ACVRL1 100.0 1000
nM
Abemaciclib ABL1(Q252H)-phosphorylated 100.0 1000
nM
Abemaciclib ABL1(F317L)-phosphorylated 100.0 100
nM
Abemaciclib AKT3 100.0 100
nM
Abemaciclib ABL1(F317L)-phosphorylated 100.0 1000
nM
Abemaciclib AKT2 100.0 100
nM
Abemaciclib CHEK1 100.0 1000
nM
Abemaciclib CDK8 100.0 100
nM