Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | AMPK-alpha2 | 100.0 | 100 | nM |
Abemaciclib | LATS1 | 100.0 | 1000 | nM |
Abemaciclib | MARK1 | 100.0 | 1000 | nM |
Abemaciclib | KIT(V559D,T670I) | 100.0 | 100 | nM |
Abemaciclib | ABL1(F317I)-phosphorylated | 100.0 | 1000 | nM |
Abemaciclib | EGFR(S752-I759del) | 100.0 | 100 | nM |
Abemaciclib | EGFR(S752-I759del) | 100.0 | 1000 | nM |
Abemaciclib | MAPKAPK5 | 100.0 | 1000 | nM |
Abemaciclib | ANKK1 | 100.0 | 100 | nM |
Abemaciclib | HCK | 100.0 | 1000 | nM |
Abemaciclib | EIF2AK1 | 100.0 | 1000 | nM |
Abemaciclib | EPHA1 | 100.0 | 100 | nM |
Abemaciclib | CDC2L1 | 100.0 | 1000 | nM |
Abemaciclib | ANKK1 | 100.0 | 1000 | nM |
Abemaciclib | CDC2L2 | 100.0 | 100 | nM |
Abemaciclib | EPHA3 | 100.0 | 100 | nM |
Abemaciclib | EPHA3 | 100.0 | 1000 | nM |
Abemaciclib | CDC2L2 | 100.0 | 1000 | nM |
Abemaciclib | EPHA4 | 100.0 | 1000 | nM |
Abemaciclib | MERTK | 100.0 | 100 | nM |
Abemaciclib | EPHA5 | 100.0 | 1000 | nM |
Abemaciclib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Abemaciclib | EPHA6 | 100.0 | 1000 | nM |
Abemaciclib | TYK2(JH2domain-pseudokinase) | 100.0 | 100 | nM |
Abemaciclib | TYK2(JH1domain-catalytic) | 100.0 | 100 | nM |