Abemaciclib KINOMEscan - Dataset (ID:20338)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Abemaciclib | EGFR(L858R) | 92.0 | 1000 | nM |
Abemaciclib | KKCC1 | 20.0 | 1000 | nM |
Abemaciclib | EGFR(L858R,T790M) | 41.0 | 1000 | nM |
Abemaciclib | MLK1 | 84.0 | 1000 | nM |
Abemaciclib | EGFR(L861Q) | 75.0 | 1000 | nM |
Abemaciclib | CAMKK2 | 4.7 | 1000 | nM |
Abemaciclib | EGFR(S752-I759del) | 100.0 | 1000 | nM |
Abemaciclib | AMPK-alpha2 | 82.0 | 1000 | nM |
Abemaciclib | EGFR(T790M) | 65.0 | 1000 | nM |
Abemaciclib | CASK | 49.0 | 1000 | nM |
Abemaciclib | EIF2AK1 | 100.0 | 1000 | nM |
Abemaciclib | ABL1-phosphorylated | 94.0 | 1000 | nM |
Abemaciclib | EPHA1 | 97.0 | 1000 | nM |
Abemaciclib | CDC2L1 | 100.0 | 1000 | nM |
Abemaciclib | EPHA2 | 94.0 | 1000 | nM |
Abemaciclib | ANKK1 | 100.0 | 1000 | nM |
Abemaciclib | EPHA3 | 100.0 | 1000 | nM |
Abemaciclib | CDC2L2 | 100.0 | 1000 | nM |
Abemaciclib | EPHA4 | 100.0 | 1000 | nM |
Abemaciclib | ABL1(H396P)-phosphorylated | 96.0 | 1000 | nM |
Abemaciclib | EPHA5 | 100.0 | 1000 | nM |
Abemaciclib | CDC2L5 | 8.0 | 1000 | nM |
Abemaciclib | EPHA6 | 100.0 | 1000 | nM |
Abemaciclib | NUAK1 | 99.0 | 1000 | nM |
Abemaciclib | MST2 | 100.0 | 1000 | nM |