Abemaciclib KINOMEscan - Dataset (ID:20338)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Abemaciclib | DMPK2 | 91.0 | 1000 | nM |
| Abemaciclib | DRAK1 | 68.0 | 100 | nM |
| Abemaciclib | DRAK1 | 1.4 | 1000 | nM |
| Abemaciclib | DRAK2 | 88.0 | 100 | nM |
| Abemaciclib | DRAK2 | 15.0 | 1000 | nM |
| Abemaciclib | DYRK1A | 2.3 | 100 | nM |
| Abemaciclib | DYRK1A | 0.0 | 1000 | nM |
| Abemaciclib | DYRK1B | 1.0 | 100 | nM |
| Abemaciclib | DYRK1B | 0.8 | 1000 | nM |
| Abemaciclib | DYRK2 | 2.8 | 100 | nM |
| Abemaciclib | DYRK2 | 0.9 | 1000 | nM |
| Abemaciclib | EGFR | 100.0 | 100 | nM |
| Abemaciclib | EGFR | 98.0 | 1000 | nM |
| Abemaciclib | EGFR(E746-A750del) | 92.0 | 100 | nM |
| Abemaciclib | EGFR(E746-A750del) | 76.0 | 1000 | nM |
| Abemaciclib | EGFR(G719C) | 86.0 | 100 | nM |
| Abemaciclib | EGFR(G719C) | 83.0 | 1000 | nM |
| Abemaciclib | EGFR(G719S) | 89.0 | 100 | nM |
| Abemaciclib | EGFR(G719S) | 84.0 | 1000 | nM |
| Abemaciclib | EGFR(L747-E749del, A750P) | 100.0 | 100 | nM |
| Abemaciclib | EGFR(L747-E749del, A750P) | 85.0 | 1000 | nM |
| Abemaciclib | EGFR(L747-S752del, P753S) | 88.0 | 100 | nM |
| Abemaciclib | EGFR(L747-S752del, P753S) | 68.0 | 1000 | nM |
| Abemaciclib | EGFR(L747-T751del,Sins) | 89.0 | 100 | nM |
| Abemaciclib | EGFR(L747-T751del,Sins) | 80.0 | 1000 | nM |