ERK5-IN-1 KINOMEscan - Dataset (ID:20337)

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Small Molecule Protein % Control Assay compound conc Conc unit
ERK5-IN-1 ABL1(F317I)-phosphorylated 64.0 1
uM
ERK5-IN-1 AURKC 66.0 1
uM
ERK5-IN-1 DYRK1B 71.0 1
uM
ERK5-IN-1 ABL1(F317L)-nonphosphorylated 71.0 1
uM
ERK5-IN-1 JNK3 74.0 1
uM
ERK5-IN-1 KIT(A829P) 74.0 1
uM
ERK5-IN-1 PIK3CA(I800L) 75.0 1
uM
ERK5-IN-1 PIK3CA(H1047Y) 76.0 1
uM
ERK5-IN-1 JNK1 76.0 1
uM
ERK5-IN-1 ROCK1 77.0 1
uM
ERK5-IN-1 FYN 78.0 1
uM
ERK5-IN-1 EGFR(L858R,T790M) 78.0 1
uM
ERK5-IN-1 TAOK2 78.0 1
uM
ERK5-IN-1 PIP5K1A 78.0 1
uM
ERK5-IN-1 CAMK2B 78.0 1
uM
ERK5-IN-1 NLK 78.0 1
uM
ERK5-IN-1 TAOK1 79.0 1
uM
ERK5-IN-1 TNK2 80.0 1
uM
ERK5-IN-1 TYK2(JH1domain-catalytic) 81.0 1
uM
ERK5-IN-1 DDR2 81.0 1
uM
ERK5-IN-1 MK11 81.0 1
uM
ERK5-IN-1 SgK110 81.0 1
uM
ERK5-IN-1 RIOK2 81.0 1
uM
ERK5-IN-1 TAOK3 82.0 1
uM
ERK5-IN-1 SRMS 82.0 1
uM