Ceritinib KINOMEscan - Dataset (ID:20329)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Ceritinib | ACVR1 | 97.0 | 1 | uM |
Ceritinib | ABL2 | 95.0 | 1 | uM |
Ceritinib | ABL1(Y253F)-phosphorylated | 65.0 | 1 | uM |
Ceritinib | ABL1(T315I)-phosphorylated | 97.0 | 1 | uM |
Ceritinib | ABL1(T315I)-nonphosphorylated | 77.0 | 1 | uM |
Ceritinib | ABL1(Q252H)-phosphorylated | 69.0 | 1 | uM |
Ceritinib | ABL1(Q252H)-nonphosphorylated | 80.0 | 1 | uM |
Ceritinib | ABL1-phosphorylated | 86.0 | 1 | uM |
Ceritinib | ABL1-nonphosphorylated | 90.0 | 1 | uM |
Ceritinib | ABL1(M351T)-phosphorylated | 100.0 | 1 | uM |
Ceritinib | ABL1(H396P)-phosphorylated | 66.0 | 1 | uM |
Ceritinib | ABL1(H396P)-nonphosphorylated | 87.0 | 1 | uM |
Ceritinib | ABL1(F317L)-phosphorylated | 35.0 | 1 | uM |
Ceritinib | ABL1(F317L)-nonphosphorylated | 50.0 | 1 | uM |
Ceritinib | ABL1(F317I)-phosphorylated | 47.0 | 1 | uM |
Ceritinib | ABL1(F317I)-nonphosphorylated | 68.0 | 1 | uM |
Ceritinib | ABL1(E255K)-phosphorylated | 70.0 | 1 | uM |
Ceritinib | AAK1 | 89.0 | 1 | uM |