Ceritinib KINOMEscan - Dataset (ID:20329)
Proteins Studied
Download: Excel (XLSX), Comma-separated (CSV)
LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200440 | TNK1 | 200440 | Q13470 | Non-receptor tyrosine-protein kinase TNK1; MGC46193; TNK1 | KINOMEscan | Wild Type; Full length | |||
200450 | TYK2(JH1domain-catalytic) | 200450 | P29597 | Non-receptor tyrosine-protein kinase TYK2; Tyrosine kinase 2; JTK1; TYK2 | KINOMEscan | JH1domain-catalytic | Wild Type; Partial length | ||
200451 | TYK2(JH2domain-pseudokinase) | 200451 | P29597 | Non-receptor tyrosine-protein kinase TYK2; Tyrosine kinase 2; JTK1; TYK2 | KINOMEscan | JH2domain-pseudokinase | Wild Type; Partial length | ||
200041 | NUAK1 | 200041 | O60285 | NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1 | KINOMEscan | Wild Type; Partial length | |||
200413 | SNARK | 200413 | Q9H093 | NUAK family, SNF1-like kinase, 2; DKFZp434J037; DKFZp686F01113; FLJ90349; NUAK2; SNARK | KINOMEscan | Wild Type; Partial length | |||
200302 | PAK1 | 200302 | Q13153 | P21 protein (Cdc42/Rac)-activated kinase 1; MGC130000; MGC130001; PAK1; PAKalpha | KINOMEscan | Wild Type; Partial length | |||
200303 | PAK2 | 200303 | Q13177 | P21 protein (Cdc42/Rac)-activated kinase 2; PAK2; PAK65; PAKgamma | KINOMEscan | Wild Type; Partial length | |||
200304 | PAK3 | 200304 | O75914 | P21 protein (Cdc42/Rac)-activated kinase 3; bPAK; CDKN1A; hPAK3; MRX30; MRX47; OPHN3; PAK3; PAK3beta | KINOMEscan | Wild Type; Full length | |||
200305 | PAK4 | 200305 | O96013 | P21 protein (Cdc42/Rac)-activated kinase 4; PAK4 | KINOMEscan | Wild Type; Partial length | |||
200306 | PAK6 | 200306 | Q9NQU5 | P21 protein (Cdc42/Rac)-activated kinase 6; PAK5; PAK6 | KINOMEscan | Wild Type; Partial length | |||
200307 | PAK7 | 200307 | Q9P286 | P21 protein (Cdc42/Rac)-activated kinase 7; KIAA1264; MGC26232; PAK5; PAK7 | KINOMEscan | Wild Type; Partial length | |||
201332 | PIK3C3 | 201332 | Q8NEB9 | Phosphatidylinositol 3-kinase catalytic subunit type 3; PI3-kinase type 3; VPS34 | KINOMEscan | ||||
200324 | PIK3CA(C420R) | 200324 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | C420R | Mutation (C420R); Partial length | ||
200332 | PIK3CA(Q546K) | 200332 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | Q546K | Mutation (Q546K); Partial length | ||
200331 | PIK3CA(M1043I) | 200331 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | M1043I | Mutation (M1043I); Partial length | ||
200330 | PIK3CA(I800L) | 200330 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | I800L | Mutation (I800L); Partial length | ||
200329 | PIK3CA(H1047Y) | 200329 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | H1047Y | Mutation (H1047Y); Partial length | ||
200323 | PIK3CA | 200323 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | Wild Type; Partial length | |||
200328 | PIK3CA(H1047L) | 200328 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | H1047L | Mutation (H1047L); Partial length | ||
200327 | PIK3CA(E545K) | 200327 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | E545K | Mutation (E545K); Partial length | ||
200326 | PIK3CA(E545A) | 200326 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | E545A | Mutation (E545A); Partial length | ||
200325 | PIK3CA(E542K) | 200325 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KINOMEscan | E542K | Mutation (E542K); Partial length | ||
200333 | PIK3CB | 200333 | P42338 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit beta; DKFZp779K1237; MGC133043; P110BETA; PI3K; PI3KBETA; PIK3C1; PIK3CB; PI3K-beta | KINOMEscan | Wild Type; Partial length | |||
200334 | PIK3CD | 200334 | O00329 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit delta; p110D; P110DELTA; PI3K; PIK3CD; PI3K-delta | KINOMEscan | Wild Type; Partial length | |||
200335 | PIK3CG | 200335 | P48736 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit gamma; PI3CG; PI3K; PI3Kgamma; PIK3; PIK3CG | KINOMEscan | Wild Type; Partial length |