Ceritinib KINOMEscan - Dataset (ID:20329)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200440 TNK1 200440 Q13470
Non-receptor tyrosine-protein kinase TNK1; MGC46193; TNK1
KINOMEscan Wild Type; Full length
200450 TYK2(JH1domain-catalytic) 200450 P29597
Non-receptor tyrosine-protein kinase TYK2; Tyrosine kinase 2; JTK1; TYK2
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200451 TYK2(JH2domain-pseudokinase) 200451 P29597
Non-receptor tyrosine-protein kinase TYK2; Tyrosine kinase 2; JTK1; TYK2
KINOMEscan JH2domain-pseudokinase Wild Type; Partial length
200041 NUAK1 200041 O60285
NUAK family, SNF1-like kinase, 1; ARK5; KIAA0537; NUAK1
KINOMEscan Wild Type; Partial length
200413 SNARK 200413 Q9H093
NUAK family, SNF1-like kinase, 2; DKFZp434J037; DKFZp686F01113; FLJ90349; NUAK2; SNARK
KINOMEscan Wild Type; Partial length
200302 PAK1 200302 Q13153
P21 protein (Cdc42/Rac)-activated kinase 1; MGC130000; MGC130001; PAK1; PAKalpha
KINOMEscan Wild Type; Partial length
200303 PAK2 200303 Q13177
P21 protein (Cdc42/Rac)-activated kinase 2; PAK2; PAK65; PAKgamma
KINOMEscan Wild Type; Partial length
200304 PAK3 200304 O75914
P21 protein (Cdc42/Rac)-activated kinase 3; bPAK; CDKN1A; hPAK3; MRX30; MRX47; OPHN3; PAK3; PAK3beta
KINOMEscan Wild Type; Full length
200305 PAK4 200305 O96013
P21 protein (Cdc42/Rac)-activated kinase 4; PAK4
KINOMEscan Wild Type; Partial length
200306 PAK6 200306 Q9NQU5
P21 protein (Cdc42/Rac)-activated kinase 6; PAK5; PAK6
KINOMEscan Wild Type; Partial length
200307 PAK7 200307 Q9P286
P21 protein (Cdc42/Rac)-activated kinase 7; KIAA1264; MGC26232; PAK5; PAK7
KINOMEscan Wild Type; Partial length
201332 PIK3C3 201332 Q8NEB9
Phosphatidylinositol 3-kinase catalytic subunit type 3; PI3-kinase type 3; VPS34
KINOMEscan
200324 PIK3CA(C420R) 200324 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan C420R Mutation (C420R); Partial length
200332 PIK3CA(Q546K) 200332 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan Q546K Mutation (Q546K); Partial length
200331 PIK3CA(M1043I) 200331 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan M1043I Mutation (M1043I); Partial length
200330 PIK3CA(I800L) 200330 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan I800L Mutation (I800L); Partial length
200329 PIK3CA(H1047Y) 200329 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan H1047Y Mutation (H1047Y); Partial length
200323 PIK3CA 200323 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan Wild Type; Partial length
200328 PIK3CA(H1047L) 200328 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan H1047L Mutation (H1047L); Partial length
200327 PIK3CA(E545K) 200327 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan E545K Mutation (E545K); Partial length
200326 PIK3CA(E545A) 200326 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan E545A Mutation (E545A); Partial length
200325 PIK3CA(E542K) 200325 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KINOMEscan E542K Mutation (E542K); Partial length
200333 PIK3CB 200333 P42338
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit beta; DKFZp779K1237; MGC133043; P110BETA; PI3K; PI3KBETA; PIK3C1; PIK3CB; PI3K-beta
KINOMEscan Wild Type; Partial length
200334 PIK3CD 200334 O00329
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit delta; p110D; P110DELTA; PI3K; PIK3CD; PI3K-delta
KINOMEscan Wild Type; Partial length
200335 PIK3CG 200335 P48736
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit gamma; PI3CG; PI3K; PI3Kgamma; PIK3; PIK3CG
KINOMEscan Wild Type; Partial length