Ceritinib KINOMEscan - Dataset (ID:20329)
Proteins Studied
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LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
201410 | CDK4 | 201410 | P11802 | Cyclin-dependent kinase 4; cell division protein kinase 4 | KINOMEscan | ||||
201334 | WNK4 | 201334 | Q96J92 | Serine/threonine-protein kinase WNK4 | KINOMEscan | ||||
201333 | WNK2 | 201333 | Q9Y3S1 | Serine/threonine-protein kinase WNK2 | KINOMEscan | ||||
201332 | PIK3C3 | 201332 | Q8NEB9 | Phosphatidylinositol 3-kinase catalytic subunit type 3; PI3-kinase type 3; VPS34 | KINOMEscan | ||||
201331 | TSSK3 | 201331 | Q96PN8 | Testis-specific serine/threonine-protein kinase 3; TSK-3 | KINOMEscan | ||||
201330 | FYV1 | 201330 | Q9Y2I7 | 1-phosphatidylinositol 3-phosphate 5-kinase; PIKfyve | KINOMEscan | ||||
201329 | BARK2 | 201329 | P35626 | Beta-adrenergic receptor kinase 2; GRK3 | KINOMEscan | ||||
201328 | BARK1 | 201328 | P25098 | Beta-adrenergic receptor kinase 1; GRK2 | KINOMEscan | ||||
201327 | FLT3(ITD,F691L) | 201327 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | ITD,F691L | |||
201326 | FLT3(ITD,D835V) | 201326 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | ITD,D835V | |||
201325 | FLT3(D835V) | 201325 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | D835V | |||
201324 | CAMK1B | 201324 | Q6P2M8 | Calcium/calmodulin-dependent protein kinase type 1B; Pregnancy up-regulated non-ubiquitously-expressed CaM kinase; CaM kinase I beta | KINOMEscan | ||||
201108 | SGK2 | 201108 | Q9HBY8 | Serine/threonine-protein kinase Sgk2; Serum/glucocorticoid-regulated kinase 2 | KINOMEscan | ||||
201107 | MAP3K14 | 201107 | Q99558 | Mitogen-activated protein kinase kinase kinase 14; NF-kappa-beta-inducing kinase; NIK | KINOMEscan | ||||
200481 | NEK10 | 200481 | Q6ZWH5 | NIMA (never in mitosis gene a)- related kinase 10 | KINOMEscan | ||||
200480 | ALK(L1196M) | 200480 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | L1196M | |||
200479 | ALK(C1156Y) | 200479 | Q9UM73 | Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK | KINOMEscan | C1156Y | |||
200478 | WNK3 | 200478 | Q9BYP7 | WNK lysine deficient protein kinase 3; PRKWNK3 | KINOMEscan | ||||
200477 | WNK1 | 200477 | Q9H4A3 | WNK lysine deficient protein kinase 1; KDP; PSK; p65; HSN2; HSAN2; PRKWNK1 | KINOMEscan | ||||
200476 | SGK1 | 200476 | O00141 | Serine/threonine-protein kinase Sgk1; serum/glucocorticoid regulated kinase 1; SGK | KINOMEscan | ||||
200475 | RSK2(Kin.Dom.2-C-terminal) | 200475 | P51812 | Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2 | KINOMEscan | Kin.Dom.2-C-terminal | |||
200474 | KIT-autoinhibited | 200474 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | ||||
200473 | HASP | 200473 | Q8TF76 | Serine/threonine-protein kinase haspin; germ cell associated 2 (haspin); GSG2; HASPIN | KINOMEscan | ||||
200472 | FLT3-autoinhibited | 200472 | P36888 | Fms-related tyrosine kinase 3; CD135; FLK2; FLK-2; FLT3; FLT-3; Ly72; STK1 | KINOMEscan | ||||
200471 | CSF1R-autoinhibited | 200471 | P07333 | Colony stimulating factor 1 receptor; CD115; C-FMS; CSF1R; CSF-1R; CSF-1-R; CSFR; FIM2; FIM-2; FMS; Fms/CSFR | KINOMEscan |