CH5424802 KINOMEscan - Dataset (ID:20326)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
CH5424802 | ACVR1 | 98.0 | 1 | uM |
CH5424802 | ABL2 | 100.0 | 1 | uM |
CH5424802 | ABL1(Y253F)-phosphorylated | 67.0 | 1 | uM |
CH5424802 | ABL1(T315I)-phosphorylated | 86.0 | 1 | uM |
CH5424802 | ABL1(T315I)-nonphosphorylated | 98.0 | 1 | uM |
CH5424802 | ABL1(Q252H)-phosphorylated | 52.0 | 1 | uM |
CH5424802 | ABL1(Q252H)-nonphosphorylated | 81.0 | 1 | uM |
CH5424802 | ABL1-phosphorylated | 73.0 | 1 | uM |
CH5424802 | ABL1-nonphosphorylated | 65.0 | 1 | uM |
CH5424802 | ABL1(M351T)-phosphorylated | 62.0 | 1 | uM |
CH5424802 | ABL1(H396P)-phosphorylated | 74.0 | 1 | uM |
CH5424802 | ABL1(H396P)-nonphosphorylated | 70.0 | 1 | uM |
CH5424802 | ABL1(F317L)-phosphorylated | 2.2 | 1 | uM |
CH5424802 | ABL1(F317L)-nonphosphorylated | 24.0 | 1 | uM |
CH5424802 | ABL1(F317I)-phosphorylated | 5.5 | 1 | uM |
CH5424802 | ABL1(F317I)-nonphosphorylated | 20.0 | 1 | uM |
CH5424802 | ABL1(E255K)-phosphorylated | 75.0 | 1 | uM |
CH5424802 | AAK1 | 72.0 | 1 | uM |