Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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WM-115 | Vemurafenib | Trametinib | PF562271 | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 1 | 1634 | 576 | 0.2587 | 0.2662 | 0.3525 | 0.3525 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2318 | 206 | 0.1255 | 0.1286 | 0.0889 | 0.0918 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 11842 | 391 | 0.6751 | 0.6666 | 0.0330 | 0.0291 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 1.0000 | 0.1000 | 1.0000 | uM | 72 | hr | 1 | 1549 | 1404 | 0.0204 | 0.0153 | 0.9064 | 0.9147 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 1 | 1677 | 174 | 0.0893 | 0.0914 | 0.1038 | 0.1080 |
A-375 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 15081 | 869 | 0.8042 | 0.8521 | 0.0576 | 0.0546 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 0.3160 | uM | 72 | hr | 1 | 1792 | 210 | 0.0940 | 0.0978 | 0.1172 | 0.1134 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 1.0000 | uM | 72 | hr | 1 | 1282 | 177 | 0.0656 | 0.0610 | 0.1381 | 0.1316 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 6910 | 334 | 0.3877 | 0.3181 | 0.0483 | 0.0472 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 3.1600 | 0.3160 | 0.3160 | uM | 72 | hr | 1 | 903 | 859 | 0.0062 | 0.0055 | 0.9513 | 0.9565 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 3.1600 | uM | 72 | hr | 1 | 1074 | 145 | 0.0552 | 0.0473 | 0.1350 | 0.1511 |
A-375 | Vemurafenib | Trametinib | Dasatinib | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 1 | 766 | 180 | 0.0377 | 0.0429 | 0.2350 | 0.2266 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 1.0000 | uM | 72 | hr | 1 | 1559 | 204 | 0.0805 | 0.0712 | 0.1309 | 0.1272 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 1 | 2074 | 218 | 0.1102 | 0.1222 | 0.1051 | 0.1075 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2621 | 258 | 0.1393 | 0.1384 | 0.0984 | 0.0909 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 4932 | 1088 | 0.5803 | 0.5134 | 0.2206 | 0.2019 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 0.3160 | uM | 72 | hr | 1 | 1508 | 137 | 0.0814 | 0.0866 | 0.0908 | 0.1048 |
A-375 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 9628 | 474 | 0.5180 | 0.5111 | 0.0492 | 0.0493 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 1.0000 | uM | 72 | hr | 1 | 1226 | 930 | 0.0447 | 0.0438 | 0.7586 | 0.7492 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 1.0000 | uM | 72 | hr | 1 | 1342 | 176 | 0.0693 | 0.0610 | 0.1311 | 0.1313 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 1 | 2168 | 357 | 0.1068 | 0.1271 | 0.1647 | 0.1561 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 3.1600 | 0.3160 | 0.3160 | uM | 72 | hr | 1 | 1779 | 195 | 0.0941 | 0.0889 | 0.1096 | 0.1191 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 3.1600 | uM | 72 | hr | 1 | 913 | 154 | 0.0451 | 0.0422 | 0.1687 | 0.1591 |
WM-115 | Vemurafenib | Trametinib | PF562271 | 1.0000 | 0.1000 | 1.0000 | uM | 72 | hr | 1 | 1582 | 791 | 0.1934 | 0.1842 | 0.5000 | 0.4768 |
WM-115 | Vemurafenib | Trametinib | PF562271 | 1.0000 | 0.1000 | 0.3160 | uM | 72 | hr | 1 | 1596 | 790 | 0.1971 | 0.1963 | 0.4950 | 0.4591 |