Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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A-375 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 17086 | 890 | 0.9165 | 1.0000 | 0.0521 | 0.0517 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2318 | 206 | 0.1255 | 0.1286 | 0.0889 | 0.0918 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 2374 | 218 | 0.1281 | 0.1286 | 0.0918 | 0.0918 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 2461 | 233 | 0.1323 | 0.1286 | 0.0947 | 0.0918 |
A-375 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 15978 | 849 | 0.9722 | 1.0000 | 0.0531 | 0.0508 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 1564 | 988 | 0.0811 | 0.0901 | 0.6317 | 0.5765 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 3 | 2578 | 300 | 0.1353 | 0.1298 | 0.1164 | 0.1284 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 3 | 2657 | 368 | 0.1360 | 0.1328 | 0.1385 | 0.1351 |
COLO 858 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 1295 | 796 | 0.0835 | 0.0919 | 0.6147 | 0.5808 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 2 | 2659 | 360 | 0.1366 | 0.1298 | 0.1354 | 0.1284 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 1 | 2285 | 305 | 0.1176 | 0.1298 | 0.1335 | 0.1284 |
COLO 858 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 7489 | 1113 | 1.0576 | 1.0000 | 0.1486 | 0.1402 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 1533 | 890 | 0.0905 | 0.0901 | 0.5806 | 0.5765 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 1 | 2074 | 218 | 0.1102 | 0.1222 | 0.1051 | 0.1075 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 2 | 2549 | 285 | 0.1345 | 0.1222 | 0.1118 | 0.1075 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 3 | 2295 | 242 | 0.1219 | 0.1222 | 0.1054 | 0.1075 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 2615 | 230 | 0.1406 | 0.1384 | 0.0880 | 0.0909 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 1452 | 751 | 0.0987 | 0.0901 | 0.5172 | 0.5765 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 2511 | 217 | 0.1352 | 0.1384 | 0.0864 | 0.0909 |
COLO 858 | Vemurafenib | Trametinib | Saracatinib | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 1 | 1023 | 943 | 0.0134 | 0.0124 | 0.9218 | 0.9350 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 3 | 1488 | 982 | 0.0712 | 0.0704 | 0.6599 | 0.6512 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 3 | 1706 | 1317 | 0.0548 | 0.0458 | 0.7720 | 0.7801 |
WM-115 | Vemurafenib | Trametinib | Dasatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2157 | 541 | 0.3789 | 0.4016 | 0.2508 | 0.2480 |
MMAC-SF | Vemurafenib | Trametinib | PF562271 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 642 | 246 | 0.3424 | 0.3170 | 0.3832 | 0.3752 |
MMAC-SF | Vemurafenib | Trametinib | PF562271 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 516 | 186 | 0.2853 | 0.3170 | 0.3605 | 0.3752 |