Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Taselisib | FGR | 90.0 | 1000 | nM |
| Taselisib | VGFR1 | 94.0 | 100 | nM |
| Taselisib | VGFR1 | 85.0 | 1000 | nM |
| Taselisib | FLT3 | 85.0 | 100 | nM |
| Taselisib | FLT3 | 78.0 | 1000 | nM |
| Taselisib | FLT3(D835H) | 92.0 | 100 | nM |
| Taselisib | FLT3(D835H) | 89.0 | 1000 | nM |
| Taselisib | FLT3(D835V) | 68.0 | 100 | nM |
| Taselisib | FLT3(D835V) | 87.0 | 1000 | nM |
| Taselisib | FLT3(D835Y) | 99.0 | 100 | nM |
| Taselisib | FLT3(D835Y) | 95.0 | 1000 | nM |
| Taselisib | FLT3(ITD) | 100.0 | 100 | nM |
| Taselisib | FLT3(ITD) | 100.0 | 1000 | nM |
| Taselisib | FLT3(ITD,D835V) | 90.0 | 100 | nM |
| Taselisib | FLT3(ITD,D835V) | 76.0 | 1000 | nM |
| Taselisib | FLT3(ITD,F691L) | 94.0 | 100 | nM |
| Taselisib | FLT3(ITD,F691L) | 93.0 | 1000 | nM |
| Taselisib | FLT3(K663Q) | 100.0 | 100 | nM |
| Taselisib | FLT3(K663Q) | 100.0 | 1000 | nM |
| Taselisib | FLT3(N841I) | 100.0 | 100 | nM |
| Taselisib | FLT3(N841I) | 100.0 | 1000 | nM |
| Taselisib | FLT3(R834Q) | 100.0 | 100 | nM |
| Taselisib | FLT3(R834Q) | 100.0 | 1000 | nM |
| Taselisib | FLT3-autoinhibited | 77.0 | 100 | nM |
| Taselisib | FLT3-autoinhibited | 89.0 | 1000 | nM |