Taselisib KINOMEscan - Dataset (ID:20264)
Proteins Studied
Download: Excel (XLSX), Comma-separated (CSV)
LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200211 | JNK1 | 200211 | P45983 | Mitogen-activated protein kinase 8; JNK; JNK1; JNK1A2; JNK21B1/2; MAPK8; PRKM8; SAPK1 | KINOMEscan | Wild Type; Full length | |||
200213 | JNK3 | 200213 | P53779 | Mitogen-activated protein kinase 10; FLJ12099; FLJ33785; JNK3; JNK3A; MAPK10; MGC50974; p493F12; p54bSAPK; PRKM10 | KINOMEscan | Wild Type; Partial length | |||
200100 | KC1G1 | 200100 | Q9HCP0 | Casein kinase I isoform gamma-1; CK1g1; CSNK1G1 | KINOMEscan | Wild Type; Partial length | |||
200101 | KC1G2 | 200101 | P78368 | Casein kinase I isoform gamma-2; Casein kinase 1, gamma 2; CK1g2; CSNK1G2 | KINOMEscan | Wild Type; Full length | |||
200065 | KCC2D | 200065 | Q13557 | Calcium/calmodulin-dependent protein kinase type II subunit delta; CaM kinase II subunit delta; CAMK2D; CAMKD; DKFZp686G23119; DKFZp686I2288; MGC44911 | KINOMEscan | Wild Type; Partial length | |||
200067 | KCC4 | 200067 | Q16566 | Calcium/calmodulin-dependent protein kinase type IV; CAMK4; CaMK-GR; MGC36771 | KINOMEscan | Wild Type; Partial length | |||
200362 | KGP1 | 200362 | Q13976 | Protein kinase, cGMP-dependent, type I; CGKI; cGKI-alpha; cGKI-BETA; DKFZp686K042; FLJ36117; MGC71944; PGK; PKG; PKG1; PRKG1; PRKG1B; PRKGR1B | KINOMEscan | Wild Type; Partial length | |||
200363 | KGP2 | 200363 | Q13237 | Protein kinase, cGMP-dependent, type II; cGKII; PKG2; PRKG2; PRKGR2 | KINOMEscan | Wild Type; Partial length | |||
200214 | KIT | 200214 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | Wild Type; Partial length | |||
200215 | KIT(A829P) | 200215 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | A829P | Mutation (A829P); Partial length | ||
200474 | KIT-autoinhibited | 200474 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | ||||
200216 | KIT(D816H) | 200216 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | D816H | Mutation (D816H); Partial length | ||
200217 | KIT(D816V) | 200217 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | D816V | Mutation (D816V); Partial length | ||
200218 | KIT(L576P) | 200218 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | L576P | Mutation (L576P); Partial length | ||
200219 | KIT(V559D) | 200219 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | V559D | Mutation (V559D); Partial length | ||
200220 | KIT(V559D,T670I) | 200220 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | V559D,T670I | Mutation (V559D,T670I); Partial length | ||
200221 | KIT(V559D,V654A) | 200221 | P10721 | V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog; CD117; C-Kit; KIT; PBT; SCFR | KINOMEscan | V559D,V654A | Mutation (V559D,V654A); Partial length | ||
200068 | KKCC1 | 200068 | Q8N5S9 | Calcium/calmodulin-dependent protein kinase kinase 1, CaM-kinase IV kinase; CAMKK1; CAMKKA; DKFZp761M0423; MGC34095 | KINOMEscan | Wild Type; Partial length | |||
200354 | KPCD | 200354 | Q05655 | Protein kinase C, delta; May1; MGC49908; nPKC-delta; PKCD; PRKCD | KINOMEscan | Wild Type; Partial length | |||
200359 | KPCD1 | 200359 | Q15139 | Protein kinase D1; PKCM; PKC-MU; PKD; PKD1; PRKCM; PRKD1 | KINOMEscan | Wild Type; Partial length | |||
200360 | KPCD2 | 200360 | Q9BZL6 | Protein kinase D2; HSPC187; PKD2; PRKD2 | KINOMEscan | Wild Type; Partial length | |||
200361 | KPCD3 | 200361 | O94806 | Protein kinase D3; EPK2; nPKC-NU; PKC-NU; PKD3; PRKCN; PRKD3 | KINOMEscan | Wild Type; Partial length | |||
200355 | KPCE | 200355 | Q02156 | Protein kinase C, epsilon; MGC125656; MGC125657; nPKC-epsilon; PKCE; PRKCE | KINOMEscan | Wild Type; Partial length | |||
200357 | KPCI | 200357 | P41743 | Protein kinase C, iota; DXS1179E; MGC26534; nPKC-iota; PKCI; PRKCI | KINOMEscan | Wild Type; Partial length | |||
200356 | KPCL | 200356 | P24723 | Protein kinase C, eta; MGC26269; MGC5363; nPKC-eta; PKCL; PKC-L; PRKCH; PRKCL | KINOMEscan | Wild Type; Partial length |