Taselisib KINOMEscan - Dataset (ID:20264)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200025 ABL1-phosphorylated 200025 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan phosphorylated Wild Type; Partial length
200024 ABL1-nonphosphorylated 200024 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan nonphosphorylated Wild Type; Partial length
200023 ABL1(Y253F)-phosphorylated 200023 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan Y253F phosphorylated Mutation (Y253F); Partial length
200021 ABL1(T315I)-phosphorylated 200021 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan T315I phosphorylated Mutation (T315I); Partial length
200020 ABL1(T315I)-nonphosphorylated 200020 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan T315I nonphosphorylated Mutation (T315I); Partial length
200018 ABL1(Q252H)-phosphorylated 200018 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan Q252H phosphorylated Mutation (Q252H); Partial length
200017 ABL1(Q252H)-nonphosphorylated 200017 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan Q252H nonphosphorylated Mutation (Q252H); Partial length
200015 ABL1(M351T)-phosphorylated 200015 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan M351T phosphorylated Mutation (M351T); Partial length
200013 ABL1(H396P)-phosphorylated 200013 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan H396P phosphorylated Mutation (H396P); Partial length
200012 ABL1(H396P)-nonphosphorylated 200012 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan H396P nonphosphorylated Mutation (H396P); Partial length
200010 ABL1(F317L)-phosphorylated 200010 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan F317L phosphorylated Mutation (F317L); Partial length
200009 ABL1(F317L)-nonphosphorylated 200009 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan F317L nonphosphorylated Mutation (F317L); Partial length
200007 ABL1(F317I)-phosphorylated 200007 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan F317I phosphorylated Mutation (F317I); Partial length
200006 ABL1(F317I)-nonphosphorylated 200006 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan F317I nonphosphorylated Mutation (F317I); Partial length
200470 BUB1 200470
Budding uninhibited by benzimidazoles 1 homolog (yeast); BUB1A; BUB1L; hBUB1
KINOMEscan
200058 BRSK2 200058 Q8IWQ3
BR serine/threonine kinase 2; BRSK2; C11orf7; FLJ41362; PEN11B; SAD1; STK29
KINOMEscan Wild Type; Full length
200057 BRSK1 200057 Q8TDC3
BR serine/threonine kinase 1; BRSK1; FLJ43009; KIAA1811
KINOMEscan Wild Type; Partial length
200052 BMPR2 200052 Q13873
Bone morphogenetic protein receptor, type II (serine/threonine kinase); BMPR2; BMPR3; BMPR-II; BMR2; BRK-3; FLJ41585; FLJ76945; PPH1; T-ALK
KINOMEscan Wild Type; Partial length
200051 BMPR1B 200051 O00238
Bone morphogenetic protein receptor, type IB; ALK6; ALK-6; BMPR1B; CDw293
KINOMEscan Wild Type; Partial length
200050 BMPR1A 200050 P36894
Bone morphogenetic protein receptor, type IA; 10q23del; ACVRLK3; ALK3; BMPR1A; CD292; SKR5
KINOMEscan Wild Type; Partial length
200053 BMX 200053 P51813
BMX non-receptor tyrosine kinase; BMX; ETK; Etk/BMX; PSCTK2; PSCTK3
KINOMEscan Wild Type; Full length
200048 BIKE 200048 Q9NSY1
BMP2 inducible kinase; BIKE; BMP2K; DKFZp434K0614; DKFZp434P0116; HRIHFB2017
KINOMEscan Wild Type; Partial length
201329 BARK2 201329 P35626
Beta-adrenergic receptor kinase 2; GRK3
KINOMEscan
201328 BARK1 201328 P25098
Beta-adrenergic receptor kinase 1; GRK2
KINOMEscan
200047 AXL 200047 P30530
AXL receptor tyrosine kinase; AXL; JTK11; UFO
KINOMEscan Wild Type; Partial length