BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib AURKB 91.0 1000
nM
Alpelisib AURKC 95.0 100
nM
Alpelisib AURKC 98.0 1000
nM
Alpelisib AXL 97.0 100
nM
Alpelisib AXL 100.0 1000
nM
Alpelisib BIKE 93.0 100
nM
Alpelisib BIKE 94.0 1000
nM
Alpelisib BLK 93.0 100
nM
Alpelisib BLK 95.0 1000
nM
Alpelisib BMPR1A 97.0 100
nM
Alpelisib BMPR1A 97.0 1000
nM
Alpelisib BMPR1B 97.0 100
nM
Alpelisib BMPR1B 98.0 1000
nM
Alpelisib BMPR2 100.0 100
nM
Alpelisib BMPR2 100.0 1000
nM
Alpelisib BMX 98.0 100
nM
Alpelisib BMX 95.0 1000
nM
Alpelisib BRAF 85.0 100
nM
Alpelisib BRAF 100.0 1000
nM
Alpelisib BRAF(V600E) 97.0 100
nM
Alpelisib BRAF(V600E) 100.0 1000
nM
Alpelisib PTK6 99.0 100
nM
Alpelisib PTK6 98.0 1000
nM
Alpelisib BRSK1 100.0 100
nM
Alpelisib BRSK1 100.0 1000
nM