BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | AURKB | 91.0 | 1000 | nM |
Alpelisib | AURKC | 95.0 | 100 | nM |
Alpelisib | AURKC | 98.0 | 1000 | nM |
Alpelisib | AXL | 97.0 | 100 | nM |
Alpelisib | AXL | 100.0 | 1000 | nM |
Alpelisib | BIKE | 93.0 | 100 | nM |
Alpelisib | BIKE | 94.0 | 1000 | nM |
Alpelisib | BLK | 93.0 | 100 | nM |
Alpelisib | BLK | 95.0 | 1000 | nM |
Alpelisib | BMPR1A | 97.0 | 100 | nM |
Alpelisib | BMPR1A | 97.0 | 1000 | nM |
Alpelisib | BMPR1B | 97.0 | 100 | nM |
Alpelisib | BMPR1B | 98.0 | 1000 | nM |
Alpelisib | BMPR2 | 100.0 | 100 | nM |
Alpelisib | BMPR2 | 100.0 | 1000 | nM |
Alpelisib | BMX | 98.0 | 100 | nM |
Alpelisib | BMX | 95.0 | 1000 | nM |
Alpelisib | BRAF | 85.0 | 100 | nM |
Alpelisib | BRAF | 100.0 | 1000 | nM |
Alpelisib | BRAF(V600E) | 97.0 | 100 | nM |
Alpelisib | BRAF(V600E) | 100.0 | 1000 | nM |
Alpelisib | PTK6 | 99.0 | 100 | nM |
Alpelisib | PTK6 | 98.0 | 1000 | nM |
Alpelisib | BRSK1 | 100.0 | 100 | nM |
Alpelisib | BRSK1 | 100.0 | 1000 | nM |