BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib TEC 99.0 100
nM
Alpelisib TEC 98.0 1000
nM
Alpelisib TESK1 91.0 100
nM
Alpelisib TESK1 88.0 1000
nM
Alpelisib TGFBR1 98.0 100
nM
Alpelisib TGFBR1 100.0 1000
nM
Alpelisib TGFBR2 96.0 100
nM
Alpelisib TGFBR2 100.0 1000
nM
Alpelisib TIE1 100.0 100
nM
Alpelisib TIE1 100.0 1000
nM
Alpelisib TIE2 96.0 100
nM
Alpelisib TIE2 89.0 1000
nM
Alpelisib TLK1 81.0 100
nM
Alpelisib TLK1 76.0 1000
nM
Alpelisib TLK2 74.0 100
nM
Alpelisib TLK2 82.0 1000
nM
Alpelisib TNIK 100.0 100
nM
Alpelisib TNIK 94.0 1000
nM
Alpelisib TNK1 84.0 100
nM
Alpelisib TNK1 67.0 1000
nM
Alpelisib TNK2 100.0 100
nM
Alpelisib TNK2 96.0 1000
nM
Alpelisib TNNI3K 99.0 100
nM
Alpelisib TNNI3K 100.0 1000
nM
Alpelisib TRKA 100.0 100
nM