BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | TEC | 99.0 | 100 | nM |
Alpelisib | TEC | 98.0 | 1000 | nM |
Alpelisib | TESK1 | 91.0 | 100 | nM |
Alpelisib | TESK1 | 88.0 | 1000 | nM |
Alpelisib | TGFBR1 | 98.0 | 100 | nM |
Alpelisib | TGFBR1 | 100.0 | 1000 | nM |
Alpelisib | TGFBR2 | 96.0 | 100 | nM |
Alpelisib | TGFBR2 | 100.0 | 1000 | nM |
Alpelisib | TIE1 | 100.0 | 100 | nM |
Alpelisib | TIE1 | 100.0 | 1000 | nM |
Alpelisib | TIE2 | 96.0 | 100 | nM |
Alpelisib | TIE2 | 89.0 | 1000 | nM |
Alpelisib | TLK1 | 81.0 | 100 | nM |
Alpelisib | TLK1 | 76.0 | 1000 | nM |
Alpelisib | TLK2 | 74.0 | 100 | nM |
Alpelisib | TLK2 | 82.0 | 1000 | nM |
Alpelisib | TNIK | 100.0 | 100 | nM |
Alpelisib | TNIK | 94.0 | 1000 | nM |
Alpelisib | TNK1 | 84.0 | 100 | nM |
Alpelisib | TNK1 | 67.0 | 1000 | nM |
Alpelisib | TNK2 | 100.0 | 100 | nM |
Alpelisib | TNK2 | 96.0 | 1000 | nM |
Alpelisib | TNNI3K | 99.0 | 100 | nM |
Alpelisib | TNNI3K | 100.0 | 1000 | nM |
Alpelisib | TRKA | 100.0 | 100 | nM |