BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Alpelisib | JNK3 | 100.0 | 1000 | nM |
| Alpelisib | KIT | 94.0 | 100 | nM |
| Alpelisib | KIT | 96.0 | 1000 | nM |
| Alpelisib | KIT(A829P) | 100.0 | 100 | nM |
| Alpelisib | KIT(A829P) | 100.0 | 1000 | nM |
| Alpelisib | KIT(D816H) | 100.0 | 100 | nM |
| Alpelisib | KIT(D816H) | 100.0 | 1000 | nM |
| Alpelisib | KIT(D816V) | 100.0 | 100 | nM |
| Alpelisib | KIT(D816V) | 100.0 | 1000 | nM |
| Alpelisib | KIT(L576P) | 81.0 | 100 | nM |
| Alpelisib | KIT(L576P) | 98.0 | 1000 | nM |
| Alpelisib | KIT(V559D) | 100.0 | 100 | nM |
| Alpelisib | KIT(V559D) | 100.0 | 1000 | nM |
| Alpelisib | KIT(V559D,T670I) | 100.0 | 100 | nM |
| Alpelisib | KIT(V559D,T670I) | 100.0 | 1000 | nM |
| Alpelisib | KIT(V559D,V654A) | 93.0 | 100 | nM |
| Alpelisib | KIT(V559D,V654A) | 100.0 | 1000 | nM |
| Alpelisib | KIT-autoinhibited | 96.0 | 100 | nM |
| Alpelisib | KIT-autoinhibited | 99.0 | 1000 | nM |
| Alpelisib | LATS1 | 94.0 | 100 | nM |
| Alpelisib | LATS1 | 83.0 | 1000 | nM |
| Alpelisib | LATS2 | 100.0 | 100 | nM |
| Alpelisib | LATS2 | 100.0 | 1000 | nM |
| Alpelisib | LCK | 65.0 | 100 | nM |
| Alpelisib | LCK | 82.0 | 1000 | nM |