BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib FLT4 100.0 100
nM
Alpelisib FLT4 100.0 1000
nM
Alpelisib FRK 93.0 100
nM
Alpelisib FRK 94.0 1000
nM
Alpelisib FYN 91.0 100
nM
Alpelisib FYN 96.0 1000
nM
Alpelisib GAK 97.0 100
nM
Alpelisib GAK 81.0 1000
nM
Alpelisib GCN2(Kin.Dom.2,S808G) 78.0 100
nM
Alpelisib GCN2(Kin.Dom.2,S808G) 78.0 1000
nM
Alpelisib GRK1 96.0 100
nM
Alpelisib GRK1 100.0 1000
nM
Alpelisib BARK1 100.0 100
nM
Alpelisib BARK1 100.0 1000
nM
Alpelisib BARK2 100.0 100
nM
Alpelisib BARK2 100.0 1000
nM
Alpelisib GRK4 92.0 100
nM
Alpelisib GRK4 90.0 1000
nM
Alpelisib GRK7 97.0 100
nM
Alpelisib GRK7 100.0 1000
nM
Alpelisib GSK3A 100.0 100
nM
Alpelisib GSK3A 82.0 1000
nM
Alpelisib GSK3B 98.0 100
nM
Alpelisib GSK3B 100.0 1000
nM
Alpelisib HASP 83.0 100
nM