BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | FLT4 | 100.0 | 100 | nM |
Alpelisib | FLT4 | 100.0 | 1000 | nM |
Alpelisib | FRK | 93.0 | 100 | nM |
Alpelisib | FRK | 94.0 | 1000 | nM |
Alpelisib | FYN | 91.0 | 100 | nM |
Alpelisib | FYN | 96.0 | 1000 | nM |
Alpelisib | GAK | 97.0 | 100 | nM |
Alpelisib | GAK | 81.0 | 1000 | nM |
Alpelisib | GCN2(Kin.Dom.2,S808G) | 78.0 | 100 | nM |
Alpelisib | GCN2(Kin.Dom.2,S808G) | 78.0 | 1000 | nM |
Alpelisib | GRK1 | 96.0 | 100 | nM |
Alpelisib | GRK1 | 100.0 | 1000 | nM |
Alpelisib | BARK1 | 100.0 | 100 | nM |
Alpelisib | BARK1 | 100.0 | 1000 | nM |
Alpelisib | BARK2 | 100.0 | 100 | nM |
Alpelisib | BARK2 | 100.0 | 1000 | nM |
Alpelisib | GRK4 | 92.0 | 100 | nM |
Alpelisib | GRK4 | 90.0 | 1000 | nM |
Alpelisib | GRK7 | 97.0 | 100 | nM |
Alpelisib | GRK7 | 100.0 | 1000 | nM |
Alpelisib | GSK3A | 100.0 | 100 | nM |
Alpelisib | GSK3A | 82.0 | 1000 | nM |
Alpelisib | GSK3B | 98.0 | 100 | nM |
Alpelisib | GSK3B | 100.0 | 1000 | nM |
Alpelisib | HASP | 83.0 | 100 | nM |