BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | DMPK2 | 100.0 | 1000 | nM |
Alpelisib | DRAK1 | 91.0 | 100 | nM |
Alpelisib | DRAK1 | 72.0 | 1000 | nM |
Alpelisib | DRAK2 | 86.0 | 100 | nM |
Alpelisib | DRAK2 | 85.0 | 1000 | nM |
Alpelisib | DYRK1A | 92.0 | 100 | nM |
Alpelisib | DYRK1A | 91.0 | 1000 | nM |
Alpelisib | DYRK1B | 54.0 | 100 | nM |
Alpelisib | DYRK1B | 45.0 | 1000 | nM |
Alpelisib | DYRK2 | 94.0 | 100 | nM |
Alpelisib | DYRK2 | 100.0 | 1000 | nM |
Alpelisib | EGFR | 97.0 | 100 | nM |
Alpelisib | EGFR | 100.0 | 1000 | nM |
Alpelisib | EGFR(E746-A750del) | 100.0 | 100 | nM |
Alpelisib | EGFR(E746-A750del) | 93.0 | 1000 | nM |
Alpelisib | EGFR(G719C) | 100.0 | 100 | nM |
Alpelisib | EGFR(G719C) | 100.0 | 1000 | nM |
Alpelisib | EGFR(G719S) | 100.0 | 100 | nM |
Alpelisib | EGFR(G719S) | 96.0 | 1000 | nM |
Alpelisib | EGFR(L747-E749del, A750P) | 99.0 | 100 | nM |
Alpelisib | EGFR(L747-E749del, A750P) | 97.0 | 1000 | nM |
Alpelisib | EGFR(L747-S752del, P753S) | 96.0 | 100 | nM |
Alpelisib | EGFR(L747-S752del, P753S) | 92.0 | 1000 | nM |
Alpelisib | EGFR(L747-T751del,Sins) | 96.0 | 100 | nM |
Alpelisib | EGFR(L747-T751del,Sins) | 78.0 | 1000 | nM |