BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib AKT2 100.0 100
nM
Alpelisib AKT2 100.0 1000
nM
Alpelisib AKT3 100.0 100
nM
Alpelisib AKT3 95.0 1000
nM
Alpelisib ALK 92.0 100
nM
Alpelisib ALK 98.0 1000
nM
Alpelisib ALK(C1156Y) 100.0 100
nM
Alpelisib ALK(C1156Y) 100.0 1000
nM
Alpelisib ALK(L1196M) 91.0 100
nM
Alpelisib ALK(L1196M) 100.0 1000
nM
Alpelisib AMPK-alpha1 88.0 100
nM
Alpelisib AMPK-alpha1 91.0 1000
nM
Alpelisib AMPK-alpha2 98.0 100
nM
Alpelisib AMPK-alpha2 100.0 1000
nM
Alpelisib ANKK1 100.0 100
nM
Alpelisib ANKK1 100.0 1000
nM
Alpelisib NUAK1 100.0 100
nM
Alpelisib NUAK1 100.0 1000
nM
Alpelisib M3K5 89.0 100
nM
Alpelisib M3K5 90.0 1000
nM
Alpelisib M3K6 100.0 100
nM
Alpelisib M3K6 100.0 1000
nM
Alpelisib AURKA 100.0 100
nM
Alpelisib AURKA 100.0 1000
nM
Alpelisib AURKB 93.0 100
nM