BYL719 KINOMEscan - Dataset (ID:20263)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | AKT2 | 100.0 | 100 | nM |
Alpelisib | AKT2 | 100.0 | 1000 | nM |
Alpelisib | AKT3 | 100.0 | 100 | nM |
Alpelisib | AKT3 | 95.0 | 1000 | nM |
Alpelisib | ALK | 92.0 | 100 | nM |
Alpelisib | ALK | 98.0 | 1000 | nM |
Alpelisib | ALK(C1156Y) | 100.0 | 100 | nM |
Alpelisib | ALK(C1156Y) | 100.0 | 1000 | nM |
Alpelisib | ALK(L1196M) | 91.0 | 100 | nM |
Alpelisib | ALK(L1196M) | 100.0 | 1000 | nM |
Alpelisib | AMPK-alpha1 | 88.0 | 100 | nM |
Alpelisib | AMPK-alpha1 | 91.0 | 1000 | nM |
Alpelisib | AMPK-alpha2 | 98.0 | 100 | nM |
Alpelisib | AMPK-alpha2 | 100.0 | 1000 | nM |
Alpelisib | ANKK1 | 100.0 | 100 | nM |
Alpelisib | ANKK1 | 100.0 | 1000 | nM |
Alpelisib | NUAK1 | 100.0 | 100 | nM |
Alpelisib | NUAK1 | 100.0 | 1000 | nM |
Alpelisib | M3K5 | 89.0 | 100 | nM |
Alpelisib | M3K5 | 90.0 | 1000 | nM |
Alpelisib | M3K6 | 100.0 | 100 | nM |
Alpelisib | M3K6 | 100.0 | 1000 | nM |
Alpelisib | AURKA | 100.0 | 100 | nM |
Alpelisib | AURKA | 100.0 | 1000 | nM |
Alpelisib | AURKB | 93.0 | 100 | nM |