BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Alpelisib | FGR | 93.0 | 1000 | nM |
| Alpelisib | VGFR1 | 88.0 | 100 | nM |
| Alpelisib | VGFR1 | 94.0 | 1000 | nM |
| Alpelisib | FLT3 | 82.0 | 100 | nM |
| Alpelisib | FLT3 | 82.0 | 1000 | nM |
| Alpelisib | FLT3(D835H) | 100.0 | 100 | nM |
| Alpelisib | FLT3(D835H) | 96.0 | 1000 | nM |
| Alpelisib | FLT3(D835V) | 100.0 | 100 | nM |
| Alpelisib | FLT3(D835V) | 82.0 | 1000 | nM |
| Alpelisib | FLT3(D835Y) | 100.0 | 100 | nM |
| Alpelisib | FLT3(D835Y) | 100.0 | 1000 | nM |
| Alpelisib | FLT3(ITD) | 100.0 | 100 | nM |
| Alpelisib | FLT3(ITD) | 100.0 | 1000 | nM |
| Alpelisib | FLT3(ITD,D835V) | 93.0 | 100 | nM |
| Alpelisib | FLT3(ITD,D835V) | 97.0 | 1000 | nM |
| Alpelisib | FLT3(ITD,F691L) | 95.0 | 100 | nM |
| Alpelisib | FLT3(ITD,F691L) | 95.0 | 1000 | nM |
| Alpelisib | FLT3(K663Q) | 100.0 | 100 | nM |
| Alpelisib | FLT3(K663Q) | 100.0 | 1000 | nM |
| Alpelisib | FLT3(N841I) | 83.0 | 100 | nM |
| Alpelisib | FLT3(N841I) | 100.0 | 1000 | nM |
| Alpelisib | FLT3(R834Q) | 100.0 | 100 | nM |
| Alpelisib | FLT3(R834Q) | 100.0 | 1000 | nM |
| Alpelisib | FLT3-autoinhibited | 98.0 | 100 | nM |
| Alpelisib | FLT3-autoinhibited | 100.0 | 1000 | nM |