Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib DYRK2 100.0 100
nM
Buparlisib EGFR 100.0 1000
nM
Buparlisib EGFR 98.0 100
nM
Buparlisib EGFR(E746-A750del) 79.0 1000
nM
Buparlisib EGFR(E746-A750del) 86.0 100
nM
Buparlisib EGFR(G719C) 98.0 100
nM
Buparlisib EGFR(G719C) 94.0 1000
nM
Buparlisib EGFR(G719S) 87.0 1000
nM
Buparlisib EGFR(G719S) 100.0 100
nM
Buparlisib EGFR(L747-E749del, A750P) 100.0 1000
nM
Buparlisib EGFR(L747-E749del, A750P) 100.0 100
nM
Buparlisib EGFR(L747-S752del, P753S) 60.0 1000
nM
Buparlisib EGFR(L747-S752del, P753S) 75.0 100
nM
Buparlisib EGFR(L747-T751del,Sins) 99.0 100
nM
Buparlisib EGFR(L747-T751del,Sins) 80.0 1000
nM
Buparlisib EGFR(L858R) 100.0 100
nM
Buparlisib EGFR(L858R) 100.0 1000
nM
Buparlisib EGFR(L858R,T790M) 100.0 1000
nM
Buparlisib EGFR(L858R,T790M) 100.0 100
nM
Buparlisib EGFR(L861Q) 69.0 1000
nM
Buparlisib EGFR(L861Q) 98.0 100
nM
Buparlisib EGFR(S752-I759del) 100.0 100
nM
Buparlisib EGFR(S752-I759del) 89.0 1000
nM
Buparlisib EGFR(T790M) 100.0 100
nM
Buparlisib EGFR(T790M) 100.0 1000
nM