Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib PIK3CG 33.0 1000
nM
Buparlisib PIK3CA(H1047L) 35.0 100
nM
Buparlisib RSK4(Kin.Dom.2-C-terminal) 37.0 100
nM
Buparlisib CLK1 47.0 1000
nM
Buparlisib DDR2 54.0 1000
nM
Buparlisib MTOR 55.0 100
nM
Buparlisib GCN2(Kin.Dom.2,S808G) 55.0 1000
nM
Buparlisib GCN2(Kin.Dom.2,S808G) 59.0 100
nM
Buparlisib EGFR(L747-S752del, P753S) 60.0 1000
nM
Buparlisib RSK2(Kin.Dom.2-C-terminal) 60.0 100
nM
Buparlisib TLK1 61.0 1000
nM
Buparlisib WEE1 62.0 1000
nM
Buparlisib CAMK1G 62.0 100
nM
Buparlisib YANK3 62.0 100
nM
Buparlisib RSK3(Kin.Dom.2-C-terminal) 62.0 1000
nM
Buparlisib RSK1(Kin.Dom.2-C-terminal) 63.0 1000
nM
Buparlisib RIOK1 63.0 100
nM
Buparlisib PIP5K1C 63.0 100
nM
Buparlisib AAK1 63.0 100
nM
Buparlisib DAPK1 64.0 1000
nM
Buparlisib TNK1 65.0 1000
nM
Buparlisib TNIK 65.0 1000
nM
Buparlisib CDKL1 67.0 100
nM
Buparlisib ABL1-nonphosphorylated 68.0 1000
nM
Buparlisib PI42C 68.0 100
nM