Buparlisib KINOMEscan - Dataset (ID:20262)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Buparlisib | PIK3CG | 33.0 | 1000 | nM |
Buparlisib | PIK3CA(H1047L) | 35.0 | 100 | nM |
Buparlisib | RSK4(Kin.Dom.2-C-terminal) | 37.0 | 100 | nM |
Buparlisib | CLK1 | 47.0 | 1000 | nM |
Buparlisib | DDR2 | 54.0 | 1000 | nM |
Buparlisib | MTOR | 55.0 | 100 | nM |
Buparlisib | GCN2(Kin.Dom.2,S808G) | 55.0 | 1000 | nM |
Buparlisib | GCN2(Kin.Dom.2,S808G) | 59.0 | 100 | nM |
Buparlisib | EGFR(L747-S752del, P753S) | 60.0 | 1000 | nM |
Buparlisib | RSK2(Kin.Dom.2-C-terminal) | 60.0 | 100 | nM |
Buparlisib | TLK1 | 61.0 | 1000 | nM |
Buparlisib | WEE1 | 62.0 | 1000 | nM |
Buparlisib | CAMK1G | 62.0 | 100 | nM |
Buparlisib | YANK3 | 62.0 | 100 | nM |
Buparlisib | RSK3(Kin.Dom.2-C-terminal) | 62.0 | 1000 | nM |
Buparlisib | RSK1(Kin.Dom.2-C-terminal) | 63.0 | 1000 | nM |
Buparlisib | RIOK1 | 63.0 | 100 | nM |
Buparlisib | PIP5K1C | 63.0 | 100 | nM |
Buparlisib | AAK1 | 63.0 | 100 | nM |
Buparlisib | DAPK1 | 64.0 | 1000 | nM |
Buparlisib | TNK1 | 65.0 | 1000 | nM |
Buparlisib | TNIK | 65.0 | 1000 | nM |
Buparlisib | CDKL1 | 67.0 | 100 | nM |
Buparlisib | ABL1-nonphosphorylated | 68.0 | 1000 | nM |
Buparlisib | PI42C | 68.0 | 100 | nM |