Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib AKT2 76.0 1000
nM
Buparlisib AKT3 100.0 100
nM
Buparlisib AKT3 94.0 1000
nM
Buparlisib ALK 82.0 100
nM
Buparlisib ALK 93.0 1000
nM
Buparlisib ALK(C1156Y) 100.0 100
nM
Buparlisib ALK(C1156Y) 100.0 1000
nM
Buparlisib ALK(L1196M) 79.0 100
nM
Buparlisib ALK(L1196M) 100.0 1000
nM
Buparlisib AMPK-alpha1 97.0 100
nM
Buparlisib AMPK-alpha1 97.0 1000
nM
Buparlisib AMPK-alpha2 100.0 100
nM
Buparlisib AMPK-alpha2 100.0 1000
nM
Buparlisib ANKK1 100.0 100
nM
Buparlisib ANKK1 100.0 1000
nM
Buparlisib NUAK1 91.0 100
nM
Buparlisib NUAK1 83.0 1000
nM
Buparlisib M3K5 91.0 100
nM
Buparlisib M3K5 100.0 1000
nM
Buparlisib M3K6 100.0 100
nM
Buparlisib M3K6 100.0 1000
nM
Buparlisib AURKA 100.0 100
nM
Buparlisib AURKA 100.0 1000
nM
Buparlisib AURKB 100.0 100
nM
Buparlisib AAK1 63.0 100
nM