Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib ABL1(Y253F)-phosphorylated 100.0 100
nM
Buparlisib ABL1(Y253F)-phosphorylated 100.0 1000
nM
Buparlisib ABL1-nonphosphorylated 94.0 100
nM
Buparlisib ABL1-nonphosphorylated 68.0 1000
nM
Buparlisib ABL1-phosphorylated 98.0 100
nM
Buparlisib ABL1-phosphorylated 100.0 1000
nM
Buparlisib ABL2 99.0 100
nM
Buparlisib ABL2 100.0 1000
nM
Buparlisib ACVR1 100.0 100
nM
Buparlisib ACVR1 100.0 1000
nM
Buparlisib ACVR1B 100.0 100
nM
Buparlisib ACVR1B 82.0 1000
nM
Buparlisib ACVR2A 95.0 100
nM
Buparlisib ACVR2A 75.0 1000
nM
Buparlisib ACVR2B 91.0 100
nM
Buparlisib ACVR2B 72.0 1000
nM
Buparlisib ACVRL1 100.0 100
nM
Buparlisib ACVRL1 99.0 1000
nM
Buparlisib ADCK3 98.0 100
nM
Buparlisib ADCK3 88.0 1000
nM
Buparlisib ADCK4 90.0 100
nM
Buparlisib ADCK4 96.0 1000
nM
Buparlisib AKT1 98.0 100
nM
Buparlisib AKT1 99.0 1000
nM
Buparlisib AAK1 63.0 100
nM