Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib AMPK-alpha2 100.0 100
nM
Buparlisib EGFR(L858R,T790M) 100.0 100
nM
Buparlisib CAMKK2 89.0 100
nM
Buparlisib EGFR(L861Q) 98.0 100
nM
Buparlisib AAK1 63.0 100
nM
Buparlisib EGFR(S752-I759del) 100.0 100
nM
Buparlisib CASK 90.0 100
nM
Buparlisib EGFR(T790M) 100.0 100
nM
Buparlisib ANKK1 100.0 100
nM
Buparlisib EIF2AK1 100.0 100
nM
Buparlisib CDC2L1 94.0 100
nM
Buparlisib EPHA1 100.0 100
nM
Buparlisib ABL2 99.0 100
nM
Buparlisib EPHA2 100.0 100
nM
Buparlisib CDC2L2 100.0 100
nM
Buparlisib EPHA3 100.0 100
nM
Buparlisib NUAK1 91.0 100
nM
Buparlisib EPHA4 98.0 100
nM
Buparlisib CDC2L5 93.0 100
nM
Buparlisib EPHA5 96.0 100
nM
Buparlisib ABL1(M351T)-phosphorylated 100.0 100
nM
Buparlisib EPHA6 93.0 100
nM
Buparlisib CDK11 100.0 100
nM
Buparlisib EPHA7 100.0 100
nM
Buparlisib MST2 99.0 100
nM