Buparlisib KINOMEscan - Dataset (ID:20262)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Buparlisib | AMPK-alpha2 | 100.0 | 100 | nM |
Buparlisib | EGFR(L858R,T790M) | 100.0 | 100 | nM |
Buparlisib | CAMKK2 | 89.0 | 100 | nM |
Buparlisib | EGFR(L861Q) | 98.0 | 100 | nM |
Buparlisib | AAK1 | 63.0 | 100 | nM |
Buparlisib | EGFR(S752-I759del) | 100.0 | 100 | nM |
Buparlisib | CASK | 90.0 | 100 | nM |
Buparlisib | EGFR(T790M) | 100.0 | 100 | nM |
Buparlisib | ANKK1 | 100.0 | 100 | nM |
Buparlisib | EIF2AK1 | 100.0 | 100 | nM |
Buparlisib | CDC2L1 | 94.0 | 100 | nM |
Buparlisib | EPHA1 | 100.0 | 100 | nM |
Buparlisib | ABL2 | 99.0 | 100 | nM |
Buparlisib | EPHA2 | 100.0 | 100 | nM |
Buparlisib | CDC2L2 | 100.0 | 100 | nM |
Buparlisib | EPHA3 | 100.0 | 100 | nM |
Buparlisib | NUAK1 | 91.0 | 100 | nM |
Buparlisib | EPHA4 | 98.0 | 100 | nM |
Buparlisib | CDC2L5 | 93.0 | 100 | nM |
Buparlisib | EPHA5 | 96.0 | 100 | nM |
Buparlisib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Buparlisib | EPHA6 | 93.0 | 100 | nM |
Buparlisib | CDK11 | 100.0 | 100 | nM |
Buparlisib | EPHA7 | 100.0 | 100 | nM |
Buparlisib | MST2 | 99.0 | 100 | nM |