Buparlisib KINOMEscan - Dataset (ID:20262)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Buparlisib | PIK3CA(H1047L) | 35.0 | 100 | nM |
Buparlisib | PIK3CA(H1047L) | 0.9 | 1000 | nM |
Buparlisib | PIK3CA(E545K) | 7.1 | 100 | nM |
Buparlisib | PIK3CA(E545K) | 0.1 | 1000 | nM |
Buparlisib | PIK3CA(E545A) | 12.0 | 100 | nM |
Buparlisib | PIK3CA(E545A) | 0.7 | 1000 | nM |
Buparlisib | PIK3CA(E542K) | 15.0 | 100 | nM |
Buparlisib | PIK3CA(E542K) | 0.3 | 1000 | nM |
Buparlisib | PIK3CA(C420R) | 0.6 | 1000 | nM |
Buparlisib | PIK3CA(C420R) | 12.0 | 100 | nM |
Buparlisib | PIK3CA | 1.4 | 1000 | nM |
Buparlisib | PIK3CA | 27.0 | 100 | nM |
Buparlisib | PIK3C3 | 14.0 | 1000 | nM |
Buparlisib | PIK3C3 | 71.0 | 100 | nM |
Buparlisib | PIK3C2G | 91.0 | 100 | nM |
Buparlisib | PIK3C2G | 69.0 | 1000 | nM |
Buparlisib | PIK3C2B | 100.0 | 100 | nM |
Buparlisib | PIK3C2B | 100.0 | 1000 | nM |
Buparlisib | PI42C | 68.0 | 100 | nM |
Buparlisib | PI42C | 79.0 | 1000 | nM |
Buparlisib | PHKG2 | 98.0 | 100 | nM |
Buparlisib | PHKG2 | 100.0 | 1000 | nM |
Buparlisib | PHKG1 | 100.0 | 100 | nM |
Buparlisib | PHKG1 | 100.0 | 1000 | nM |
Buparlisib | PGFRB | 100.0 | 100 | nM |