Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib PIK3CA(H1047L) 35.0 100
nM
Buparlisib PIK3CA(H1047L) 0.9 1000
nM
Buparlisib PIK3CA(E545K) 7.1 100
nM
Buparlisib PIK3CA(E545K) 0.1 1000
nM
Buparlisib PIK3CA(E545A) 12.0 100
nM
Buparlisib PIK3CA(E545A) 0.7 1000
nM
Buparlisib PIK3CA(E542K) 15.0 100
nM
Buparlisib PIK3CA(E542K) 0.3 1000
nM
Buparlisib PIK3CA(C420R) 0.6 1000
nM
Buparlisib PIK3CA(C420R) 12.0 100
nM
Buparlisib PIK3CA 1.4 1000
nM
Buparlisib PIK3CA 27.0 100
nM
Buparlisib PIK3C3 14.0 1000
nM
Buparlisib PIK3C3 71.0 100
nM
Buparlisib PIK3C2G 91.0 100
nM
Buparlisib PIK3C2G 69.0 1000
nM
Buparlisib PIK3C2B 100.0 100
nM
Buparlisib PIK3C2B 100.0 1000
nM
Buparlisib PI42C 68.0 100
nM
Buparlisib PI42C 79.0 1000
nM
Buparlisib PHKG2 98.0 100
nM
Buparlisib PHKG2 100.0 1000
nM
Buparlisib PHKG1 100.0 100
nM
Buparlisib PHKG1 100.0 1000
nM
Buparlisib PGFRB 100.0 100
nM