Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib CDK7 98.0 100
nM
Buparlisib CDK7 100.0 1000
nM
Buparlisib CDK8 86.0 100
nM
Buparlisib CDK8 77.0 1000
nM
Buparlisib CDK9 82.0 100
nM
Buparlisib CDK9 91.0 1000
nM
Buparlisib CDKL1 67.0 100
nM
Buparlisib CDKL1 88.0 1000
nM
Buparlisib CDKL2 94.0 100
nM
Buparlisib CDKL2 89.0 1000
nM
Buparlisib CDKL3 99.0 100
nM
Buparlisib CDKL3 99.0 1000
nM
Buparlisib CDKL5 100.0 100
nM
Buparlisib CDKL5 97.0 1000
nM
Buparlisib CHEK1 100.0 100
nM
Buparlisib CHEK1 100.0 1000
nM
Buparlisib CHK2 100.0 100
nM
Buparlisib CHK2 100.0 1000
nM
Buparlisib CIT 97.0 100
nM
Buparlisib CIT 100.0 1000
nM
Buparlisib CLK1 98.0 100
nM
Buparlisib CLK1 47.0 1000
nM
Buparlisib CLK2 89.0 100
nM
Buparlisib CLK2 98.0 1000
nM
Buparlisib CLK3 100.0 100
nM