Buparlisib KINOMEscan - Dataset (ID:20262)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200024 ABL1-nonphosphorylated 200024 P00519
C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl
KINOMEscan nonphosphorylated Wild Type; Partial length
200038 AMPK-alpha1 200038 Q13131
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPKa1; AMPK-alpha1; MGC33776; MGC57364; PRKAA1
KINOMEscan Wild Type; Partial length
200037 ALK 200037 Q9UM73
Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK
KINOMEscan Wild Type; Partial length
200039 AMPK-alpha2 200039 P54646
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPK2; AMPKa2; AMPK-alpha2; PRKAA; PRKAA2
KINOMEscan Wild Type; Partial length
200040 ANKK1 200040 Q8NFD2
Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288
KINOMEscan Wild Type; Partial length
200063 CAMK2A 200063 Q9UQM7
Calcium/calmodulin-dependent protein kinase II alpha; CAMK2A; CAMKA; KIAA0968
KINOMEscan Wild Type; Partial length
200070 CASK 200070 O14936
Calcium/calmodulin-dependent serine protein kinase (MAGUK family); CAGH39; CAMGUK; CASK; CMG; FGS4; FLJ22219; FLJ31914; LIN2; MICPCH; TNRC8
KINOMEscan Wild Type; Partial length
200036 AKT3 200036 Q9Y243
V-akt murine thymoma viral oncogene homolog 3 (protein kinase B, gamma); AKT3; Akt3/PKBg; DKFZp434N0250; PKBg; PKB-GAMMA; PRKBG; RAC-gamma; RAC-PK-gamma; STK-2
KINOMEscan Wild Type; Partial length
200035 AKT2 200035 P31751
V-akt murine thymoma viral oncogene homolog 2; AKT2; Akt2/PKBb; PKBb; PKBBETA; PRKBB; RAC-BETA
KINOMEscan Wild Type; Partial length
200065 KCC2D 200065 Q13557
Calcium/calmodulin-dependent protein kinase type II subunit delta; CaM kinase II subunit delta; CAMK2D; CAMKD; DKFZp686G23119; DKFZp686I2288; MGC44911
KINOMEscan Wild Type; Partial length
200072 CDC2L2 200072 Q9UQ88
Cyclin-dependent kinase 11A; CDC2L2; CDC2L3; CDK11A; CDK11-p110; CDK11-p46; CDK11-p58; MGC131975; p58GTA; PITSLRE
KINOMEscan Wild Type; Partial length
200069 CAMKK2 200069 Q96RR4
Calcium/calmodulin-dependent protein kinase kinase 2, beta; CAMKK; CAMKK2; CAMKKB; KIAA0787; MGC15254
KINOMEscan Wild Type; Partial length
200085 CDKL3 200085 Q8IVW4
Cyclin-dependent kinase-like 3; CDKL3; NKIAMRE
KINOMEscan Wild Type; Partial length
200086 CDKL5 200086 O76039
Cyclin-dependent kinase-like 5; CDKL5; ISSX; STK9
KINOMEscan Wild Type; Partial length
200087 CHEK1 200087 O14757
CHK1 checkpoint homolog (S. pombe); CHEK1; CHK1
KINOMEscan Wild Type; Partial length
200073 CDC2L5 200073 Q14004
Cyclin-dependent kinase 13; CDC2L; CDC2L5; CDK13; CHED; FLJ35215; KIAA1791
KINOMEscan Wild Type; Partial length
200054 BRAF 200054 P15056
Serine/threonine-protein kinase B-raf; v-raf murine sarcoma viral oncogene homolog B1; BRAF1; RAFB1
KINOMEscan Wild Type; Partial length
200031 ACVRL1 200031 P37023
Activin A receptor type II-like 1; ACVRL1; ACVRLK1; ALK1; ALK-1; HHT; HHT2; ORW2; SKR3; TSR-I
KINOMEscan Wild Type; Partial length
200067 KCC4 200067 Q16566
Calcium/calmodulin-dependent protein kinase type IV; CAMK4; CaMK-GR; MGC36771
KINOMEscan Wild Type; Partial length
200066 CAMK2G 200066 Q13555
Calcium/calmodulin-dependent protein kinase II gamma; CAMK; CAMK2G; CAMKG; CAMK-II; FLJ16043; MGC26678
KINOMEscan Wild Type; Partial length
200056 PTK6 200056 Q13882
Protein tyrosine kinase 6; BRK; FLJ42088; PTK6
KINOMEscan Wild Type; Partial length
200057 BRSK1 200057 Q8TDC3
BR serine/threonine kinase 1; BRSK1; FLJ43009; KIAA1811
KINOMEscan Wild Type; Partial length
200061 CAMK1D 200061 Q8IU85
Calcium/calmodulin-dependent protein kinase ID; CaM-K1; CAMK1D; CaMKID; CKLiK
KINOMEscan Wild Type; Partial length
200074 CDK11 200074 Q9BWU1
Cyclin-dependent kinase 19; bA346C16.3; CDC2L6; CDK11; CDK19; KIAA1028
KINOMEscan Wild Type; Partial length
200052 BMPR2 200052 Q13873
Bone morphogenetic protein receptor, type II (serine/threonine kinase); BMPR2; BMPR3; BMPR-II; BMR2; BRK-3; FLJ41585; FLJ76945; PPH1; T-ALK
KINOMEscan Wild Type; Partial length