GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Pictilisib | CDK7 | 100.0 | 100 | nM |
Pictilisib | CDK7 | 100.0 | 1000 | nM |
Pictilisib | CDK8 | 90.0 | 100 | nM |
Pictilisib | CDK8 | 92.0 | 1000 | nM |
Pictilisib | CDK9 | 100.0 | 100 | nM |
Pictilisib | CDK9 | 100.0 | 1000 | nM |
Pictilisib | CDKL1 | 75.0 | 100 | nM |
Pictilisib | CDKL1 | 84.0 | 1000 | nM |
Pictilisib | CDKL2 | 95.0 | 100 | nM |
Pictilisib | CDKL2 | 92.0 | 1000 | nM |
Pictilisib | CDKL3 | 95.0 | 100 | nM |
Pictilisib | CDKL3 | 100.0 | 1000 | nM |
Pictilisib | CDKL5 | 100.0 | 100 | nM |
Pictilisib | CDKL5 | 100.0 | 1000 | nM |
Pictilisib | CHEK1 | 100.0 | 100 | nM |
Pictilisib | CHEK1 | 100.0 | 1000 | nM |
Pictilisib | CHK2 | 100.0 | 100 | nM |
Pictilisib | CHK2 | 100.0 | 1000 | nM |
Pictilisib | CIT | 97.0 | 100 | nM |
Pictilisib | CIT | 98.0 | 1000 | nM |
Pictilisib | CLK1 | 86.0 | 100 | nM |
Pictilisib | CLK1 | 59.0 | 1000 | nM |
Pictilisib | CLK2 | 99.0 | 100 | nM |
Pictilisib | CLK2 | 55.0 | 1000 | nM |
Pictilisib | CLK3 | 100.0 | 100 | nM |