GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Pictilisib | PIK3CA(C420R) | 1.9 | 100 | nM |
| Pictilisib | PIK3CA(C420R) | 0.0 | 1000 | nM |
| Pictilisib | PIK3CA(E542K) | 1.2 | 100 | nM |
| Pictilisib | PIK3CA(E542K) | 0.0 | 1000 | nM |
| Pictilisib | PIK3CA(E545A) | 1.6 | 100 | nM |
| Pictilisib | PIK3CA(E545A) | 0.0 | 1000 | nM |
| Pictilisib | PIK3CA(E545K) | 0.8 | 100 | nM |
| Pictilisib | PIK3CA(E545K) | 0.0 | 1000 | nM |
| Pictilisib | PIK3CA(H1047L) | 17.0 | 100 | nM |
| Pictilisib | PIK3CA(H1047L) | 0.8 | 1000 | nM |
| Pictilisib | PIK3CA(H1047Y) | 1.0 | 100 | nM |
| Pictilisib | PIK3CA(H1047Y) | 0.0 | 1000 | nM |
| Pictilisib | PIK3CA(I800L) | 7.0 | 100 | nM |
| Pictilisib | PIK3CA(I800L) | 0.0 | 1000 | nM |
| Pictilisib | PIK3CA(M1043I) | 0.0 | 100 | nM |
| Pictilisib | PIK3CA(M1043I) | 0.4 | 1000 | nM |
| Pictilisib | PIK3CA(Q546K) | 4.0 | 100 | nM |
| Pictilisib | PIK3CA(Q546K) | 0.1 | 1000 | nM |
| Pictilisib | PIK3CB | 15.0 | 100 | nM |
| Pictilisib | PIK3CB | 0.0 | 1000 | nM |
| Pictilisib | PIK3CD | 7.0 | 100 | nM |
| Pictilisib | PIK3CD | 0.0 | 1000 | nM |
| Pictilisib | PIK3CG | 48.0 | 100 | nM |
| Pictilisib | PIK3CG | 3.5 | 1000 | nM |
| Pictilisib | PIK4CB | 100.0 | 100 | nM |