GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Pictilisib | FGR | 100.0 | 1000 | nM |
| Pictilisib | VGFR1 | 96.0 | 100 | nM |
| Pictilisib | VGFR1 | 100.0 | 1000 | nM |
| Pictilisib | FLT3 | 91.0 | 100 | nM |
| Pictilisib | FLT3 | 67.0 | 1000 | nM |
| Pictilisib | FLT3(D835H) | 99.0 | 100 | nM |
| Pictilisib | FLT3(D835H) | 79.0 | 1000 | nM |
| Pictilisib | FLT3(D835V) | 86.0 | 100 | nM |
| Pictilisib | FLT3(D835V) | 62.0 | 1000 | nM |
| Pictilisib | FLT3(D835Y) | 100.0 | 100 | nM |
| Pictilisib | FLT3(D835Y) | 89.0 | 1000 | nM |
| Pictilisib | FLT3(ITD) | 100.0 | 100 | nM |
| Pictilisib | FLT3(ITD) | 79.0 | 1000 | nM |
| Pictilisib | FLT3(ITD,D835V) | 78.0 | 100 | nM |
| Pictilisib | FLT3(ITD,D835V) | 67.0 | 1000 | nM |
| Pictilisib | FLT3(ITD,F691L) | 92.0 | 100 | nM |
| Pictilisib | FLT3(ITD,F691L) | 71.0 | 1000 | nM |
| Pictilisib | FLT3(K663Q) | 100.0 | 100 | nM |
| Pictilisib | FLT3(K663Q) | 100.0 | 1000 | nM |
| Pictilisib | FLT3(N841I) | 100.0 | 100 | nM |
| Pictilisib | FLT3(N841I) | 100.0 | 1000 | nM |
| Pictilisib | FLT3(R834Q) | 100.0 | 100 | nM |
| Pictilisib | FLT3(R834Q) | 100.0 | 1000 | nM |
| Pictilisib | FLT3-autoinhibited | 97.0 | 100 | nM |
| Pictilisib | FLT3-autoinhibited | 100.0 | 1000 | nM |