GDC-0941 KINOMEscan-3 - Dataset (ID:20261)

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Small Molecule Protein % Control Assay compound conc Conc unit
Pictilisib PIK3CB 15.0 100
nM
Pictilisib PIK3C2G 17.0 1000
nM
Pictilisib PIK3CA(H1047L) 17.0 100
nM
Pictilisib PIK3C2B 18.0 1000
nM
Pictilisib JAK1(JH2domain-pseudokinase) 18.0 1000
nM
Pictilisib RSK2(Kin.Dom.2-C-terminal) 48.0 100
nM
Pictilisib PIK3CG 48.0 100
nM
Pictilisib PIP5K1C 51.0 100
nM
Pictilisib MYLK4 52.0 1000
nM
Pictilisib VRK2 54.0 1000
nM
Pictilisib CLK2 55.0 1000
nM
Pictilisib CLK4 56.0 1000
nM
Pictilisib EPHB6 57.0 1000
nM
Pictilisib HASP 59.0 1000
nM
Pictilisib MK12 59.0 1000
nM
Pictilisib CLK1 59.0 1000
nM
Pictilisib FYV1 59.0 100
nM
Pictilisib MKNK1 60.0 100
nM
Pictilisib HIPK2 61.0 1000
nM
Pictilisib FLT3(D835V) 62.0 1000
nM
Pictilisib CDC2L5 63.0 100
nM
Pictilisib TNIK 64.0 100
nM
Pictilisib MLK3 64.0 100
nM
Pictilisib EGFR(L747-S752del, P753S) 64.0 100
nM
Pictilisib KGP1 65.0 1000
nM