GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Pictilisib | RET | 91.0 | 1000 | nM |
| Pictilisib | FYN | 91.0 | 1000 | nM |
| Pictilisib | RIPK1 | 91.0 | 1000 | nM |
| Pictilisib | PLK1 | 91.0 | 100 | nM |
| Pictilisib | PLK1 | 91.0 | 1000 | nM |
| Pictilisib | FLT3 | 91.0 | 100 | nM |
| Pictilisib | PAK1 | 91.0 | 100 | nM |
| Pictilisib | EGFR(S752-I759del) | 91.0 | 100 | nM |
| Pictilisib | MET(Y1235D) | 92.0 | 100 | nM |
| Pictilisib | KGP1 | 92.0 | 100 | nM |
| Pictilisib | LKB1 | 92.0 | 100 | nM |
| Pictilisib | KC1G2 | 92.0 | 100 | nM |
| Pictilisib | BRAF | 92.0 | 1000 | nM |
| Pictilisib | JAK3(JH1domain-catalytic) | 92.0 | 100 | nM |
| Pictilisib | JAK1(JH1domain-catalytic) | 92.0 | 1000 | nM |
| Pictilisib | CDKL2 | 92.0 | 1000 | nM |
| Pictilisib | CDK8 | 92.0 | 1000 | nM |
| Pictilisib | FLT3(ITD,F691L) | 92.0 | 100 | nM |
| Pictilisib | ERBB2 | 92.0 | 1000 | nM |
| Pictilisib | NEK1 | 92.0 | 1000 | nM |
| Pictilisib | EGFR(G719S) | 93.0 | 1000 | nM |
| Pictilisib | KGP2 | 93.0 | 100 | nM |
| Pictilisib | MP2K7 | 93.0 | 100 | nM |
| Pictilisib | DDR2 | 93.0 | 100 | nM |
| Pictilisib | LOK | 93.0 | 1000 | nM |