GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Pictilisib | AMPK-alpha2 | 100.0 | 100 | nM |
Pictilisib | EGFR(L858R,T790M) | 98.0 | 100 | nM |
Pictilisib | CAMKK2 | 91.0 | 100 | nM |
Pictilisib | EGFR(L861Q) | 88.0 | 100 | nM |
Pictilisib | AAK1 | 89.0 | 100 | nM |
Pictilisib | EGFR(S752-I759del) | 91.0 | 100 | nM |
Pictilisib | CASK | 68.0 | 100 | nM |
Pictilisib | EGFR(T790M) | 100.0 | 100 | nM |
Pictilisib | ANKK1 | 100.0 | 100 | nM |
Pictilisib | EIF2AK1 | 100.0 | 100 | nM |
Pictilisib | CDC2L1 | 100.0 | 100 | nM |
Pictilisib | EPHA1 | 100.0 | 100 | nM |
Pictilisib | ABL2 | 100.0 | 100 | nM |
Pictilisib | EPHA2 | 77.0 | 100 | nM |
Pictilisib | CDC2L2 | 100.0 | 100 | nM |
Pictilisib | EPHA3 | 100.0 | 100 | nM |
Pictilisib | NUAK1 | 100.0 | 100 | nM |
Pictilisib | EPHA4 | 100.0 | 100 | nM |
Pictilisib | CDC2L5 | 63.0 | 100 | nM |
Pictilisib | EPHA5 | 83.0 | 100 | nM |
Pictilisib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Pictilisib | EPHA6 | 100.0 | 100 | nM |
Pictilisib | CDK11 | 100.0 | 100 | nM |
Pictilisib | EPHA7 | 100.0 | 100 | nM |
Pictilisib | MST2 | 90.0 | 100 | nM |