GDC-0941 KINOMEscan-3 - Dataset (ID:20261)

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Small Molecule Protein % Control Assay compound conc Conc unit
Pictilisib AMPK-alpha2 100.0 100
nM
Pictilisib EGFR(L858R,T790M) 98.0 100
nM
Pictilisib CAMKK2 91.0 100
nM
Pictilisib EGFR(L861Q) 88.0 100
nM
Pictilisib AAK1 89.0 100
nM
Pictilisib EGFR(S752-I759del) 91.0 100
nM
Pictilisib CASK 68.0 100
nM
Pictilisib EGFR(T790M) 100.0 100
nM
Pictilisib ANKK1 100.0 100
nM
Pictilisib EIF2AK1 100.0 100
nM
Pictilisib CDC2L1 100.0 100
nM
Pictilisib EPHA1 100.0 100
nM
Pictilisib ABL2 100.0 100
nM
Pictilisib EPHA2 77.0 100
nM
Pictilisib CDC2L2 100.0 100
nM
Pictilisib EPHA3 100.0 100
nM
Pictilisib NUAK1 100.0 100
nM
Pictilisib EPHA4 100.0 100
nM
Pictilisib CDC2L5 63.0 100
nM
Pictilisib EPHA5 83.0 100
nM
Pictilisib ABL1(M351T)-phosphorylated 100.0 100
nM
Pictilisib EPHA6 100.0 100
nM
Pictilisib CDK11 100.0 100
nM
Pictilisib EPHA7 100.0 100
nM
Pictilisib MST2 90.0 100
nM