GDC-0941 KINOMEscan-3 - Dataset (ID:20261)

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Small Molecule Protein % Control Assay compound conc Conc unit
Pictilisib EGFR(L858R) 100.0 1000
nM
Pictilisib AMPK-alpha2 100.0 100
nM
Pictilisib EGFR(L858R,T790M) 100.0 1000
nM
Pictilisib FES 100.0 1000
nM
Pictilisib AMPK-alpha2 100.0 1000
nM
Pictilisib ABL1(F317I)-phosphorylated 100.0 1000
nM
Pictilisib ABL1(H396P)-phosphorylated 100.0 1000
nM
Pictilisib EGFR(T790M) 100.0 100
nM
Pictilisib EGFR(T790M) 100.0 1000
nM
Pictilisib EIF2AK1 100.0 100
nM
Pictilisib EIF2AK1 100.0 1000
nM
Pictilisib EPHA1 100.0 100
nM
Pictilisib EPHA1 100.0 1000
nM
Pictilisib CDC2L1 100.0 1000
nM
Pictilisib CDC2L2 100.0 100
nM
Pictilisib EPHA3 100.0 100
nM
Pictilisib EPHA3 100.0 1000
nM
Pictilisib EPHA4 100.0 100
nM
Pictilisib EPHA4 100.0 1000
nM
Pictilisib NUAK1 100.0 100
nM
Pictilisib ABL1(M351T)-phosphorylated 100.0 100
nM
Pictilisib EPHA6 100.0 100
nM
Pictilisib EPHA6 100.0 1000
nM
Pictilisib EPHA7 100.0 100
nM
Pictilisib MET(M1250T) 100.0 1000
nM