GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Pictilisib | EGFR(L858R) | 100.0 | 1000 | nM |
Pictilisib | AMPK-alpha2 | 100.0 | 100 | nM |
Pictilisib | EGFR(L858R,T790M) | 100.0 | 1000 | nM |
Pictilisib | FES | 100.0 | 1000 | nM |
Pictilisib | AMPK-alpha2 | 100.0 | 1000 | nM |
Pictilisib | ABL1(F317I)-phosphorylated | 100.0 | 1000 | nM |
Pictilisib | ABL1(H396P)-phosphorylated | 100.0 | 1000 | nM |
Pictilisib | EGFR(T790M) | 100.0 | 100 | nM |
Pictilisib | EGFR(T790M) | 100.0 | 1000 | nM |
Pictilisib | EIF2AK1 | 100.0 | 100 | nM |
Pictilisib | EIF2AK1 | 100.0 | 1000 | nM |
Pictilisib | EPHA1 | 100.0 | 100 | nM |
Pictilisib | EPHA1 | 100.0 | 1000 | nM |
Pictilisib | CDC2L1 | 100.0 | 1000 | nM |
Pictilisib | CDC2L2 | 100.0 | 100 | nM |
Pictilisib | EPHA3 | 100.0 | 100 | nM |
Pictilisib | EPHA3 | 100.0 | 1000 | nM |
Pictilisib | EPHA4 | 100.0 | 100 | nM |
Pictilisib | EPHA4 | 100.0 | 1000 | nM |
Pictilisib | NUAK1 | 100.0 | 100 | nM |
Pictilisib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Pictilisib | EPHA6 | 100.0 | 100 | nM |
Pictilisib | EPHA6 | 100.0 | 1000 | nM |
Pictilisib | EPHA7 | 100.0 | 100 | nM |
Pictilisib | MET(M1250T) | 100.0 | 1000 | nM |