GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Pictilisib | EGFR(L858R) | 100.0 | 1000 | nM |
Pictilisib | KKCC1 | 84.0 | 1000 | nM |
Pictilisib | EGFR(L858R,T790M) | 100.0 | 1000 | nM |
Pictilisib | MLK1 | 100.0 | 1000 | nM |
Pictilisib | EGFR(L861Q) | 77.0 | 1000 | nM |
Pictilisib | CAMKK2 | 97.0 | 1000 | nM |
Pictilisib | EGFR(S752-I759del) | 94.0 | 1000 | nM |
Pictilisib | AMPK-alpha2 | 100.0 | 1000 | nM |
Pictilisib | EGFR(T790M) | 100.0 | 1000 | nM |
Pictilisib | CASK | 78.0 | 1000 | nM |
Pictilisib | EIF2AK1 | 100.0 | 1000 | nM |
Pictilisib | ABL1-phosphorylated | 99.0 | 1000 | nM |
Pictilisib | EPHA1 | 100.0 | 1000 | nM |
Pictilisib | CDC2L1 | 100.0 | 1000 | nM |
Pictilisib | EPHA2 | 83.0 | 1000 | nM |
Pictilisib | ANKK1 | 100.0 | 1000 | nM |
Pictilisib | EPHA3 | 100.0 | 1000 | nM |
Pictilisib | CDC2L2 | 100.0 | 1000 | nM |
Pictilisib | EPHA4 | 100.0 | 1000 | nM |
Pictilisib | ABL1(H396P)-phosphorylated | 100.0 | 1000 | nM |
Pictilisib | EPHA5 | 97.0 | 1000 | nM |
Pictilisib | CDC2L5 | 99.0 | 1000 | nM |
Pictilisib | EPHA6 | 100.0 | 1000 | nM |
Pictilisib | NUAK1 | 97.0 | 1000 | nM |
Pictilisib | MST2 | 100.0 | 1000 | nM |