GDC-0941 KINOMEscan-3 - Dataset (ID:20261)

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Small Molecule Protein % Control Assay compound conc Conc unit
Pictilisib EGFR(L858R) 100.0 1000
nM
Pictilisib KKCC1 84.0 1000
nM
Pictilisib EGFR(L858R,T790M) 100.0 1000
nM
Pictilisib MLK1 100.0 1000
nM
Pictilisib EGFR(L861Q) 77.0 1000
nM
Pictilisib CAMKK2 97.0 1000
nM
Pictilisib EGFR(S752-I759del) 94.0 1000
nM
Pictilisib AMPK-alpha2 100.0 1000
nM
Pictilisib EGFR(T790M) 100.0 1000
nM
Pictilisib CASK 78.0 1000
nM
Pictilisib EIF2AK1 100.0 1000
nM
Pictilisib ABL1-phosphorylated 99.0 1000
nM
Pictilisib EPHA1 100.0 1000
nM
Pictilisib CDC2L1 100.0 1000
nM
Pictilisib EPHA2 83.0 1000
nM
Pictilisib ANKK1 100.0 1000
nM
Pictilisib EPHA3 100.0 1000
nM
Pictilisib CDC2L2 100.0 1000
nM
Pictilisib EPHA4 100.0 1000
nM
Pictilisib ABL1(H396P)-phosphorylated 100.0 1000
nM
Pictilisib EPHA5 97.0 1000
nM
Pictilisib CDC2L5 99.0 1000
nM
Pictilisib EPHA6 100.0 1000
nM
Pictilisib NUAK1 97.0 1000
nM
Pictilisib MST2 100.0 1000
nM