Breast Cancer Cell Density: Imaging assay of the density- and context-dependence of small molecule perturbagen response in breast cancer cell lines. Dataset 3 of 3: Calculated dose-response metrics. - Dataset (ID:20258)

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Cell Small Molecule Replicate Seeding Density IC50 EC50 Emax Einf IC Hill Coefficient IC_AUC IC Curve Fit IC r2 GR50 GEC50 GRmax GRinf GR Hill Coefficient GR_AOC GR Curve Fit GR r2
MDA-MB-231 Omipalisib 11 156.25
0.1358
0.0594
0.2740 0.2830 1.0087 0.5821
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9607
0.0375
0.0462
-0.1059 -0.0926 0.8136 0.6658
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.948
MDA-MB-231 Omipalisib 11 312.50
0.1027
0.0479
0.2070 0.2144 0.7347 0.5282
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9914
0.0491
0.0704
-0.1012 -0.1199 0.5964 0.6228
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9889
MDA-MB-231 Omipalisib 11 625.00
0.0659
0.0296
0.2185 0.2365 0.8015 0.5000
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9889
0.0302
0.0357
-0.0810 -0.0599 0.6764 0.6668
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.99
MDA-MB-231 Omipalisib 11 1250.00
0.0759
0.0313
0.2166 0.2306 0.6989 0.5049
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9864
0.0335
0.0414
-0.0702 -0.0663 0.5890 0.6491
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.978
MDA-MB-231 Omipalisib 11 2500.00
0.1448
0.0411
0.2689 0.2424 0.5267 0.5418
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9975
0.0325
0.0481
-0.0623 -0.1074 0.4971 0.6514
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9939
MDA-MB-231 Omipalisib 11 5000.00
1.5766
0.5936
0.3697 0.1486 0.3610 0.6706
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9957
0.1077
0.7877
-0.2338 -0.6482 0.4177 0.5832
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9938
BT-20 NVP-TAE684 3 156.25
4.8641
2.9659
0.3686 0.3105 1.9617 0.9242
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9744
2.3148
3.1061
-0.2096 -0.3536 1.8191 0.1687
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9919
BT-20 NVP-TAE684 3 312.50
3.7935
2.1702
0.3887 0.3767 2.5072 0.9225
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9697
1.9558
2.2149
-0.1500 -0.1775 2.4417 0.1730
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9903
BT-20 NVP-TAE684 3 625.00
2.9826
2.4087
0.2572 0.2501 3.2454 0.9075
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9802
2.2539
2.5629
-0.2412 -0.2565 3.2228 0.1669
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9919
BT-20 NVP-TAE684 3 1250.00
2.4485
1.7399
0.3578 0.3576 3.6764 0.9045
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9769
1.8738
1.8372
0.0359 0.0345 3.6151 0.1553
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.989
BT-20 NVP-TAE684 3 2500.00
2.5949
1.8812
0.3282 0.3263 3.2875 0.8988
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9809
1.954
1.997
-0.0315 -0.0365 3.2405 0.1638
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.991
BT-20 NVP-TAE684 3 5000.00
3.4169
2.2807
0.3655 0.3594 3.1387 0.9070
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9858
2.2559
2.3698
-0.0710 -0.0830 3.1156 0.1609
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9937
BT-20 PLX-4720 3 156.25
23.4882
23.4881
0.6867 0.0000 5.0000 1.0144
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.8645
19.1631
23.872
0.4111 -1.0000 5.0000 0.0034
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9432
BT-20 PLX-4720 3 312.50
24.832
24.8319
0.7435 0.0000 5.0000 1.0365
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.7551
20.3724
25.3785
0.5302 -1.0000 5.0000 -0.0293
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9073
BT-20 PLX-4720 3 625.00
27.1685
27.1647
0.8198 0.0004 5.0000 1.0403
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.5695
23.3287
29.055
0.7300 -0.9984 5.0000 -0.0373
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.7686
BT-20 PLX-4720 3 1250.00
27.4271
27.4199
0.8264 0.0007 5.0000 1.0383
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.5656
24.1694
30.0978
0.7686 -0.9973 5.0000 -0.0371
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.7165
BT-20 PLX-4720 3 2500.00
inf
17.7176
0.7649 0.6333 4.7685 1.0173
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.8524
26.7937
19.9517
0.6797 0.3633 4.3971 -0.0162
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9014
BT-20 PLX-4720 3 5000.00
inf
10.2702
0.7747 0.7666 4.9996 1.0098
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.8661
inf
10.3841
0.6474 0.6340 5.0000 -0.0059
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9152
BT-20 Palbociclib 3 156.25
26.2184
26.2184
0.5812 0.0000 1.4198 0.9376
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.8603
11.6786
23.4356
0.1132 -1.0000 1.5773 0.1274
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.8903
BT-20 Palbociclib 3 312.50
inf
0.1305
0.5804 0.6126 1.8634 0.7943
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9551
0.3282
0.183
0.2493 0.2802 1.4064 0.3669
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9706
BT-20 Palbociclib 3 625.00
inf
0.0375
0.5123 0.6394 1.6869 0.7255
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.6093
0.0394
0.0262
0.1837 0.4346 5.0000 0.4701
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.5401
BT-20 Palbociclib 3 1250.00
1.0299
0.2199
0.3688 0.3792 0.9199 0.6834
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9547
0.2257
0.2381
-0.0304 -0.0221 0.8106 0.5158
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9614
BT-20 Palbociclib 3 2500.00
0.8767
0.2413
0.3802 0.3855 1.1424 0.6849
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9943
0.3481
0.2763
0.1045 0.1147 1.1275 0.4411
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9925
BT-20 Palbociclib 3 5000.00
inf
0.1503
0.5045 0.5000 0.9422 0.7166
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.9475
0.2708
0.1658
0.1953 0.1879 0.9611 0.4532
sigmoidal fit: x = Einf + (1-Einf)/(1+ (x/EC50)^Hill)
0.95
BT-20 Nilotinib 3 156.25
inf
inf
1.0500 1.0500 0.0000 0.9620
flat fit: x = Einf
0.0745
inf
inf
1.0500 1.0500 0.0000 0.0953
flat fit: x = Einf
0.0963