WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 53.1 | 1 | uM |
| WZ3105 | THP-1 | AMPKa1,AMPKa2 | VAVKILNR | Lys1 | 4.8 | 1 | uM |
| WZ3105 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | -3.8 | 1 | uM |
| WZ3105 | THP-1 | ATM | QLVKGRDDLRQDAVMQQVFQMCNTLLQR | ATP | -6.1 | 1 | uM |
| WZ3105 | THP-1 | ATR | FYIMMCKPK | ATP | 2.4 | 1 | uM |
| WZ3105 | THP-1 | AurA | FILALKVLFK | Lys1 | 4.0 | 1 | uM |
| WZ3105 | THP-1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -1.5 | 1 | uM |
| WZ3105 | THP-1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 17.1 | 1 | uM |
| WZ3105 | THP-1 | CaMK1a | LVAIKCIAK | Lys1 | 0.1 | 1 | uM |
| WZ3105 | THP-1 | CAMK1D | LFAVKCIPK | Lys1 | -2.1 | 1 | uM |
| WZ3105 | THP-1 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLKPENLLLASK | Lys2 | 27.6 | 1 | uM |
| WZ3105 | THP-1 | KCC2D | IPTGQEYAAKIINTK | Lys1 | 32.5 | 1 | uM |
| WZ3105 | THP-1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 46.3 | 1 | uM |
| WZ3105 | THP-1 | CaMKK2 | LAYNENDNTYYAMKVLSK | Lys1 | 65.2 | 1 | uM |
| WZ3105 | THP-1 | CDK20 | DLKPANLLISASGQLK | Lys2 | 4.9 | 1 | uM |
| WZ3105 | THP-1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -1.9 | 1 | uM |
| WZ3105 | THP-1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -16.9 | 1 | uM |
| WZ3105 | THP-1 | CDK2 | NKLTGEVVALKK | Lys1 | 0.6 | 1 | uM |
| WZ3105 | THP-1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 14.4 | 1 | uM |
| WZ3105 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -3.4 | 1 | uM |
| WZ3105 | THP-1 | CDK5 | NRETHEIVALKR | Lys1 | 35.7 | 1 | uM |
| WZ3105 | THP-1 | CDK5 | DLKPQNLLINR | Lys2 | 39.1 | 1 | uM |
| WZ3105 | THP-1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -2.1 | 1 | uM |
| WZ3105 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 64.4 | 1 | uM |
| WZ3105 | THP-1 | CDK9 | DMKAANVLITR | Lys2 | 23.4 | 1 | uM |