WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | CDK20 | DLKPANLLISASGQLK | Lys2 | 4.9 | 1 | uM |
| WZ3105 | THP-1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 50.1 | 1 | uM |
| WZ3105 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -3.4 | 1 | uM |
| WZ3105 | THP-1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -5.9 | 1 | uM |
| WZ3105 | THP-1 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLKPENLLLASK | Lys2 | 27.6 | 1 | uM |
| WZ3105 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | -3.8 | 1 | uM |
| WZ3105 | THP-1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | -0.8 | 1 | uM |
| WZ3105 | THP-1 | SNRK | DLKPENVVFFEK | Lys2 | -6.1 | 1 | uM |
| WZ3105 | THP-1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -12.9 | 1 | uM |
| WZ3105 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 64.4 | 1 | uM |
| WZ3105 | THP-1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -11.4 | 1 | uM |
| WZ3105 | THP-1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -2.1 | 1 | uM |
| WZ3105 | THP-1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -1.9 | 1 | uM |
| WZ3105 | THP-1 | PCTAIRE2 | DLKPQNLLINEK | Lys2 | -3.8 | 1 | uM |
| WZ3105 | THP-1 | CDK16 | DLKPQNLLINER | Lys2 | 6.7 | 1 | uM |
| WZ3105 | THP-1 | CDK5 | DLKPQNLLINR | Lys2 | 39.1 | 1 | uM |
| WZ3105 | THP-1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 14.4 | 1 | uM |
| WZ3105 | THP-1 | PKR | DLKPSNIFLVDTK | Lys2 | 3.9 | 1 | uM |
| WZ3105 | THP-1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | -12.3 | 1 | uM |
| WZ3105 | THP-1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | -10.3 | 1 | uM |
| WZ3105 | THP-1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 12.9 | 1 | uM |
| WZ3105 | THP-1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | -10.4 | 1 | uM |
| WZ3105 | THP-1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | -5.7 | 1 | uM |
| WZ3105 | THP-1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -28.5 | 1 | uM |
| WZ3105 | THP-1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -1.5 | 1 | uM |